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3-methyl-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
7-[(8-fluoro-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
[(2S,6S)-4-[(2-chloro-6-fluorophenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,2-dimethyl-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxamide
3-butyl-4-[2-(4-fluorophenyl)benzoyl]-1-methylpiperazin-2-one
methyl 6-[3-(4-fluorophenyl)pyrrolidin-1-yl]pyrimidine-4-carboxylate
methyl 1-[(3-methoxyphenyl)methoxy]-2-oxo-8-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
8-fluoro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]quinoline-2-carboxamide
3-[2-(4-methoxyphenyl)ethyl]-5-methyl-5-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
1-[6-(benzyloxy)-4-(2-methylpropyl)-3-oxo-1,4-diazepan-1-yl]-2-phenylethane-1,2-dione
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
1-{1'-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1-[({[3-(pyrrolidin-1-yl)phenyl]methyl}carbamoyl)methyl]piperidine-4-carboxamide
2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(propan-2-yl)acetamide
4-[1-(3-fluorophenyl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]pyridazine
3-(pentan-2-yl)-8-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N,N-dimethyl-5-{[(5-methylfuran-2-yl)methyl]amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
(2S,4R)-4-{[(2,6-difluorophenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)pyrrolidine-2-carboxamide
2-[2-(methylsulfanyl)ethyl]-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
4-[(3,5-dimethoxyphenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
3-[2-fluoro-3-(pyrrolidin-1-ylmethyl)phenoxy]-6-phenylpyridazine
N-ethyl-N-(oxolan-2-ylmethyl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
7-(5-methylthiophen-2-yl)-4-(pyrrolidine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-({5-[3-(3-methoxypropyl)piperidine-1-carbonyl]furan-2-yl}methyl)-4-methylpiperazine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methyl-1H-pyrazole-5-carboxamide
N-(1-{1-[(2R)-2-amino-3-methylbutanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
1-(cyclohex-3-ene-1-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-1-(propan-2-yl)piperidine-3-carboxamide
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-(pyrrolidin-1-yl)piperidin-3-yl]propan-1-one
2-amino-4-(2-methoxypyrimidin-5-yl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-methyl-1-(pyrimidin-2-yl)-N-(1,3-thiazol-2-ylmethyl)piperidin-4-amine
2-chloro-N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]pyridine-4-carboxamide
N-[3-(benzylsulfanyl)propyl]-2-(methylamino)pyridine-4-carboxamide
N-(5-methyl-4H-1,2,4-triazol-3-yl)-3-(morpholine-4-carbonyl)piperidine-1-carboxamide
2-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
8-[(4-acetylphenyl)methyl]-2-(3-hydroxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(2-{[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N,3-dimethyl-N-[(5-methylfuran-2-yl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
2-{N-methyl-1-[2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazol-4-yl]formamido}propanamide
N-{5-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]quinolin-8-yl}acetamide
6-[(4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]quinoline
1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(4aR,8aR)-7-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[4-(2-fluoro-4,5-dimethoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
1-{6-methyl-3-[(4-methyl-1,4-diazepan-1-yl)methyl]quinolin-2-yl}piperidin-3-ol
8-({4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}methyl)-2,8-diazaspiro[4.5]decan-3-one
5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-7H-[1,3]thiazolo[3,2-a]pyrimidin-7-one