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4,4-dibenzyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(2-aminopyrimidin-4-yl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
2-amino-4-(4-hydroxyphenyl)-6-[4-(morpholin-4-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
4-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
1-methyl-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}imidazolidin-2-one
2-{[4-(2-fluoro-4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-4-methylphenol
3-ethyl-6-{3-[(4-fluorophenyl)methoxy]azetidine-1-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
2-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-methoxypyrazine
{1-[({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]cyclobutyl}methanol
(3S,5R)-1-[(4-methylphenyl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-{[1-(1H-indol-2-ylmethyl)pyrrolidin-3-yl]methyl}cyclohexanecarboxamide
2-(6-chloro-2H-1,3-benzodioxol-5-yl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
N-(5-{2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetamido}-2-methylphenyl)-4-methylbenzamide
N-(4-methoxy-2-methylphenyl)-3-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)propanamide
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
2-amino-6-cyclobutyl-4-(6-methoxy-2H-1,3-benzodioxol-5-yl)pyridine-3-carbonitrile
5-[(6,8-dimethyl-4-oxo-1,4-dihydroquinolin-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-hydroxyacetamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-amine
(2R,3R,6R)-5-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1-{[1-(propan-2-yl)piperidin-4-yl]methyl}pyrrolidin-3-yl)methyl]azetidine-3-carboxamide
1-(4-methyl-1,4-diazepane-1-carbonyl)-6-[(3-phenoxyphenyl)methyl]-6-azaspiro[2.5]octane
4-{4-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]phenyl}but-3-yn-1-ol
methyl 2-(azocane-1-sulfonyl)-6-(oxolane-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(4-methylpiperazin-1-yl)-3-(4-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}phenoxy)propan-2-ol
5-{2-[(thiolan-3-yl)amino]ethyl}-1,3,4-thiadiazol-2-amine
(3aS,6aS)-2-(5-cyanopyridin-2-yl)-5-cyclopentanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
N-(5-chloro-2-methoxyphenyl)-3-[1-(pyrazin-2-yl)piperidin-3-yl]propanamide
N-cyclopentyl-4-{1,8-dioxa-4,11-diazaspiro[5.6]dodecan-4-yl}-4-oxobutanamide
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-[3-({3-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
N-(1-{7-[2-(4-acetylphenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-2-(dimethylamino)acetamide
2-(1-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-4-yl)-1,3-benzoxazole
4-{[(4aR,8aR)-7-(dimethylsulfamoyl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]methyl}benzoic acid
8-{2-[benzyl(methyl)amino]acetyl}-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N3-cyclohexyl-1-(2-methylpropyl)-4-oxo-N5-[(3S)-2-oxoazepan-3-yl]-1,4-dihydropyridine-3,5-dicarboxamide
(1R,5R)-N,N-dimethyl-6-{[4-(propan-2-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-benzyl-N-(2-hydroxyethyl)acetamide
3-(2-methylphenyl)-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}pyrrolidin-3-ol
2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(1H-pyrazol-1-yl)propanamide
N-cyclopropyl-1-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}piperidine-3-carboxamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methylpyrazolo[1,5-a]pyridine-7-carboxamide
2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
(1S,5R)-3-(2H-1,3-benzodioxol-5-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
3-{[2-(1-benzothiophen-2-yl)-1H-imidazol-1-yl]methyl}-5-(methoxymethyl)-1,2,4-oxadiazole
ethyl 2-{4-[(2E)-2-methylbut-2-en-1-yl]piperazin-1-yl}pyridine-3-carboxylate