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(3S,9aR)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
ethyl 4-benzyl-1-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}piperidine-4-carboxylate
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[2-(pyridin-4-ylformamido)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
6-methyl-4-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-2,3-dihydropyridazin-3-one
N3-(1,3-benzothiazol-2-ylmethyl)-N5-tert-butyl-N3-methyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(cyclohexylmethyl)-3-(pyridin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(3-ethoxy-4-{furo[3,2-c]pyridin-4-yloxy}phenyl)methyl]pyrrolidine
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-(2-methylphenyl)-4-{1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}piperazine
(4aS,8aR)-1-(3-methoxypropyl)-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-decahydro-1,6-naphthyridin-2-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-acetamidopropanamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-(3,3-diphenylpropyl)-6-[(4-hydroxy-3-methoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(1-benzofuran-2-ylmethyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-(4-fluorophenyl)-2-methyl-4-{1-[(2,4,6-trimethoxyphenyl)methyl]piperidin-3-yl}pyrimidine
(2,4,6-trimethyl-3-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}phenyl)methanol
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxyethan-1-one
4-[(2,3-difluorophenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(2,4-dichlorophenoxy)-N-methylacetamide
2-cyclopropyl-N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-4-methylpyrimidine-5-carboxamide
4-methyl-2-[1-(6-methylpyridazin-3-yl)piperidin-3-yl]-1H-1,3-benzodiazole
1-[4-(4-acetyl-4-phenylpiperidine-1-carbonyl)-3,5-dimethyl-1H-pyrrol-2-yl]ethan-1-one
1-{4-[3-(4-methylphenoxymethyl)piperidin-1-yl]-4-oxobutyl}pyrrolidin-2-one
2-methyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(4H-1,2,4-triazol-4-yl)pyridine
3-propyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-pyrazole-5-carboxamide
2-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N5-[(1-benzylpyrrolidin-3-yl)methyl]-N6-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
3-{2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}quinoline
1-[(5-methoxy-1,3,4-thiadiazol-2-yl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
[(3R,4R)-1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-ethyl-N-(2-hydroxyethyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-{1-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]piperidin-3-yl}acetamide
(4aR,7aS)-4-(6-aminopyridine-3-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-{4-[2-(2-methoxy-4-methylphenoxy)ethyl]piperazin-1-yl}-1,3-benzoxazole
1-(3-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propyl)piperidine-3-carboxamide
[(3R,4R)-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-(furan-2-ylmethyl)-3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-[(5-methylpyrazin-2-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-1,4-dithiepan-6-amine
N'-(5-chloro-2-methylphenyl)-N-{[1-(ethoxymethyl)cyclobutyl]methyl}propanediamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-2-methoxyacetamide
9-(3-methoxy-2-methylbenzoyl)-3-oxa-9-azaspiro[5.5]undecane
methyl 3-(oxolane-2-amido)-1-(2-phenylethyl)-5-[(1,3-thiazol-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-{1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-3-carbonyl}pyridine
3-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
1-{[4-(1,2-oxazinane-2-carbonyl)-1,3-oxazol-2-yl]methyl}-1H-1,3-benzodiazole
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-2-(3,4,5-trimethoxyphenyl)acetamide
1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole