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4-(quinoxalin-2-yl)-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[4-(benzyloxy)butyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[2-(diethylamino)pyridin-3-yl]methyl}-4-oxo-3,4-dihydrophthalazine-1-carboxamide
(4aS,8aR)-6-(2-cyclopentylacetyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
2-(1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
N-ethyl-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(pyrrolidin-1-yl)ethyl]butanamide
1-(2-methoxy-5-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
3-(azocane-1-sulfonyl)-N-[2-(propan-2-yloxy)ethyl]benzamide
5-(phenoxymethyl)-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
1'-(1,3-benzothiazole-6-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-methoxypropanamide
3-[2-(5-acetylthiophen-3-yl)acetamido]-N-(1,3-thiazol-2-yl)propanamide
2-[2-(3,4-dimethoxyphenyl)ethyl]-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-[(4-methylphenyl)methyl]-11-{[2-(pyridin-3-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2-chloro-4-fluorophenyl)-6-(piperidine-1-carbonyl)pyrazine
N-[(4-hydroxyphenyl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-({1-[(4-chloro-3-fluorophenyl)methyl]piperidin-2-yl}methyl)morpholine
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[2-(thiophen-2-yl)ethyl]azepan-4-amine
N-(4-{[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]methyl}phenyl)acetamide
1-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-(pyrrolidin-1-yl)ethan-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(4-hydroxypiperidin-1-yl)pyridine-3-carboxamide
(3R,4R)-1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-methyl-2-{2-[(2E)-2-methylbut-2-en-1-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1H-1,3-benzodiazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
N-methyl-1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]pyrrolidine-3-carboxamide
8-methoxy-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{4-[(dimethylamino)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-[2-(4-methoxyphenyl)ethyl]-2-(morpholin-4-ylmethyl)piperidine-1-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
N-methyl-1-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-(1-methylpyrrolidin-3-yl)-1,2-oxazole-3-carboxamide
3-[5-(3-fluoro-5-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
3-(azepane-1-carbonyl)-N-butyl-N-methyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-[1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
(4aR,7aS)-1-(2-methylpropyl)-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
1-(diethylamino)-3-[2-methoxy-5-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
1-cyclopentyl-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
(2E)-3-(2-chlorophenyl)-1-[4-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
9-[2-(3,4-dimethylphenoxy)ethyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrazine
3-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}pyridin-2-amine
N3-cycloheptyl-1-cyclopropyl-N5-[(3,4-dimethoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-cycloheptyl-1-cyclopropyl-5-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[(2,3-difluorophenyl)methyl]-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
1-(4-cyano-2-fluorophenyl)-3-[3-(methylsulfanyl)propyl]urea
N-(1-{7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide