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2-[N-(3-methylphenyl)methanesulfonamido]-N-[1-(thiophen-2-yl)propyl]acetamide
dimethyl(3-{2-[1-(2-methylpyrimidine-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
5-{[2-(furan-2-yl)azepan-1-yl]methyl}-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
4-[({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}carbamoyl)amino]-N,3-dimethylbenzamide
2-(4-chloro-1H-pyrazol-1-yl)-1-{2,7-diazaspiro[4.5]decan-2-yl}ethan-1-one
2-(2-methoxyethyl)-8-(4,4,4-trifluorobutanoyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(2-{[2-(dimethylamino)-2,3-dihydro-1H-inden-2-yl]formamido}ethyl)acetamide
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-1-(thiomorpholin-4-yl)propan-1-one
1-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-3-methoxypropan-1-one
2-cyclopropyl-8-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-5-(pyridin-3-yl)imidazolidine-2,4-dione
4-[4-(5,6,7,8-tetrahydro-1,6-naphthyridin-6-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
N-(2-{2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}ethyl)-1,9-dioxaspiro[5.5]undecan-4-amine
2-(1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1,3-benzoxazole
N-{1-[1-(dimethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
3-{4-[2-(4-methylpentyl)morpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}propan-1-amine
2-(2-{1-[5-(4-methylphenyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}ethyl)pyridine
1-(1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N,N,5-trimethylpyrimidin-4-amine
1-cyclobutanecarbonyl-4-(pyrimidin-4-yl)-1,4-diazepane
(4aR,7aS)-1-(2-methylpropyl)-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-4-methyl-1H-imidazole-2-carboxamide
2-{4-[(3-chlorophenyl)methyl]-1-cyclopentylpiperazin-2-yl}ethan-1-ol
4-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)piperidine-4-carboxamide
2-(2-methylpropyl)-6-[(2S)-oxolane-2-carbonyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
2-{2-[methyl(quinolin-5-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
(4aR,7aS)-1-[2-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1-{7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[2-(oxan-2-yl)ethyl]-1H-pyrazole-3-carboxamide
N,1,3,6-tetramethyl-N-[(3-methylpyridin-2-yl)methyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
7-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]acetamide
2-(1-methylpyrrolidin-3-yl)-9-(pyridazin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]butanamide
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]cyclopentanamine
3-(3-methoxyphenyl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazole-5-carboxamide
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,6-dimethylpyrimidin-4-amine
4-(3-fluoropropyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-(hydroxymethyl)-1-[(5-phenylthiophen-2-yl)methyl]azepan-4-ol
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-methyl-N-[(5-{[(2-methylpropyl)[(3-methylthiophen-2-yl)methyl]amino]methyl}furan-2-yl)methyl]methanesulfonamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(1-ethylcyclopropyl)piperidine-3-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[1-(hydroxymethyl)cyclobutyl]methyl}-5-methylpiperidin-2-one
2-[(2-phenoxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid