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4-cyclopentyl-7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}(methyl){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
N-[4-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenyl]acetamide
2-[(4aR,7aS)-4-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
7-[(4-methyl-1H-imidazol-5-yl)methyl]-N-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(2,6-dimethylpyridin-4-yl)piperazine
4-[(4-fluorophenyl)methyl]-1-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidine
4-(3-hydroxy-3-methylbutyl)-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]benzamide
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
2-({4-[6-(piperidin-1-yl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4-(1H-pyrazol-4-yl)butanamide
1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]-2-(4-phenylphenyl)ethan-1-one
5-(3,4-dimethylphenoxymethyl)-N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)-1,2-oxazole-3-carboxamide
N,1-dimethyl-5-[(2-methylpropyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,4R)-3-cyclobutyl-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-methylpyrrolidin-3-ol
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-methyl-4-(2-methylphenyl)piperazine
2-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]-1,3-thiazole
4-[6-oxo-4-(piperidin-1-yl)-1,6-dihydropyridazin-1-yl]butanamide
2-[1-(3-methylbutyl)-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl]ethan-1-ol
5-ethyl-2-methyl-4-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyrimidine
3-{[3-(3-fluoro-4-methoxybenzoyl)piperidin-1-yl]methyl}phenol
(3aR,7aS)-2-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)propanamide
2-(dimethylamino)-N-[2-(ethylsulfanyl)ethyl]-2-(3-methylphenyl)acetamide
(1R,9S)-5-amino-12-cyclopentyl-3-(pyridin-4-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
N-(5-chloro-2-methoxyphenyl)-3-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
2-[(4-benzylpiperazin-1-yl)methyl]-N-(oxan-4-ylmethyl)-1,3-oxazole-4-carboxamide
3-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)-6-methyl-1,2-dihydroquinolin-2-one
(4aR,8aS)-6-[(4-ethoxyphenyl)methyl]-1-{[4-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
1-(3-{3-[(4-fluoropiperidin-1-yl)methyl]phenoxy}-2-hydroxypropyl)piperidin-4-ol
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-[2-(2-fluorophenyl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-N-ethyl-4-{[(3-methylphenyl)methyl]amino}-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
5-[1-(2-methoxyphenyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]-2-methylpyrimidine
(4aS,7aR)-1-(2,8-dimethylquinoline-3-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{4-[3-(pyridin-4-yl)azetidine-1-carbonyl]phenyl}methanol
1-{4-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
methyl 2-({2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}methyl)-1,3-oxazole-4-carboxylate
(2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-8-methylquinolin-3-yl)methanol
1'-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}spiro[indene-1,4'-piperidine]
1-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-2-hydroxyethan-1-one
1-[(3-fluorophenyl)methyl]-4-{[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}pyrrolidin-2-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
3-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethoxy}-4-methyl-1,2,5-oxadiazole
2-{1-[(4-ethoxyphenyl)methyl]-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
4-[(oxan-4-yl)sulfamoyl]-N-(oxolan-3-yl)benzamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,1-dimethyl-1H-indole-3-carboxamide
3-[1-(3-methylbenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one