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N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-{3-[3-(6-methylpyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}-1-(piperidin-1-yl)ethan-1-one
1-(2-aminopyrimidin-4-yl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
(4aS,7aR)-1-(3-phenylpropyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-tert-butyl-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-methyl-3-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}-1,4-dihydroquinolin-4-one
N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}-2-(2-oxopiperidin-1-yl)acetamide
methyl 1-oxo-2-(oxolan-2-ylmethyl)-1,2-dihydroisoquinoline-7-carboxylate
N-benzyl-N-butyl-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-(3-methoxypropyl)-1-methyl-N-[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]piperidin-4-amine
N-(3-methoxyphenyl)-4-[2-(phenylcarbamoyl)ethyl]piperidine-1-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
N-(2-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
5-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-cyclohexyl-5-(3-ethyl-1,2-oxazol-5-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazole
2-(5-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
2-tert-butyl-N-[3-(1,3-oxazol-5-yl)phenyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
2,3-difluoro-5-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenol
1-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]-3-phenylpropan-2-ol
3-{2-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-oxoethyl}-5,5-dimethyl-1,3-oxazolidine-2,4-dione
8-(oxan-4-yl)-1-(2-phenylethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1R,3S)-7-[(3-fluoro-4-methoxyphenyl)methyl]-7-azaspiro[3.5]nonane-1,3-diol
2-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)benzonitrile
1-(4-ethylpiperazin-1-yl)-3-[3-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
2-[3-(4-methylphenoxymethyl)piperidin-1-yl]pyridine-4-carboxamide
4-(4-methanesulfonylphenyl)-6-(trifluoromethyl)-1H-1,3-benzodiazole
N-(3-chloro-4-propoxyphenyl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
2-methyl-5-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]phenol
4-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
5-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyridine-2,4-diol
[4-(8-chloroquinoline-2-carbonyl)-1,4-oxazepan-6-yl]methanol
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazole
2-(prop-2-en-1-yl)-9-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-(5-{3,9-diazaspiro[5.6]dodecan-9-ylmethyl}thiophen-3-yl)prop-2-yn-1-ol
N-({5-[(5-cyclopentylthiophen-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-{4-[(2,6-difluorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
3,5-dimethyl-1-[1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)pyrrolidin-3-yl]-1H-pyrazole
2-(1-methylcyclopentanecarbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-(methoxymethyl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidin-4-amine
4-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
N-methyl-2-[4-(propan-2-yl)morpholin-2-yl]-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
(3S,4R)-1-{[3-(2-aminoethyl)phenyl]methyl}-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
[(2S,6S)-4-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2-fluorophenyl)ethan-1-one
6-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(3S,4R)-1-({4-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide