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N-[(6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-3-yl)methyl]acetamide
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-(6-oxopiperidine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(3-oxo-2,3-dihydro-1,2-benzothiazol-2-yl)acetamide
3-[1-(6-methylquinoline-4-carbonyl)piperidin-3-yl]-1-(pyrrolidin-1-yl)propan-1-one
2-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-1,2-oxazinane
N-(2-hydroxyethyl)-N-(3-methyl-1,1-dioxo-1λ6-thiolan-3-yl)-4-(5-methylfuran-2-yl)benzamide
4-(1-methyl-1H-imidazol-2-yl)-1-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-1H-1,2,3-triazole
N-[2-(ethylsulfanyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-methyl-1-[2-(5-methylfuran-2-yl)phenyl]-3-(oxolan-3-ylmethyl)urea
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-6-(methoxymethyl)pyrimidin-4-amine
4-fluoro-N-(2-{[3-(1H-pyrazol-1-yl)phenyl]formamido}ethyl)benzamide
4-ethyl-3-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
1-(3-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-5-(5-methylthiophen-2-yl)phenyl)-1H-1,2,3,4-tetrazole
N-(2-methoxy-5-methylphenyl)-3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carboxamide
7-(2,6-dimethoxyphenyl)-4-[(3-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1-methylimidazolidin-2-one
3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-(pyridin-4-yl)ethyl]urea
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
2-cyclopropyl-8-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-N-[3-(1H-imidazol-1-yl)propyl]-2,3-dihydro-1H-indene-2-carboxamide
4-[4-(4-methoxyphenyl)-5-methyl-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
1-[3-(benzyloxy)piperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
N-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
(1S,5R)-3-benzoyl-6-(2,5-dimethylfuran-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[1-(4-methylphenyl)-5-[(4-oxo-3,4-dihydroquinazolin-3-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[3-(1H-imidazol-1-yl)propyl]propanamide
1-(4-benzylpiperidin-1-yl)-3-[1-(piperidin-4-yl)piperidin-4-yl]propan-1-one
2-(butan-2-ylsulfanyl)-5-{[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyrimidine
2-{[4-(3-acetylphenyl)phenyl]sulfanyl}acetamide
2-(4-methoxyphenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
1-(3-methoxypropyl)-5-methyl-5-phenylpiperidin-2-one
1'-(2H-1,3-benzodioxol-5-ylmethyl)-5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-(2-methoxybenzoyl)piperazine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]acetamide
5-butyl-1'-(dimethyl-1,3-oxazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{[4-(1-benzyl-1H-pyrazole-4-carbonyl)-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl]oxy}-N,N-diethylacetamide
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2,1,3-benzothiadiazole-4-sulfonamide
(1S,5R)-6-(2-methoxyethyl)-3-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
[(8-methoxy-2H-chromen-3-yl)methyl][2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]amine
2,4-dimethoxy-N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
3-(1-benzothiophen-2-ylmethyl)-3,4-dihydropteridin-4-one
(3S,4R)-1-[(2-chloro-3,6-difluorophenyl)methyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
3-{[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
3-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
2-[(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)methyl]-1,3-benzothiazole
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide