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1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(piperidin-1-yl)piperidine-4-carboxamide
N-[(1-ethylpiperidin-3-yl)methyl]-2-methyl-2-phenylpropanamide
N-(1-{7-[(4-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)furan-3-carboxamide
2-chloro-4-({[2-(1-hydroxycyclopentyl)ethyl](methyl)carbamoyl}amino)benzamide
ethyl 4-[3-({[(3-fluorophenyl)methyl]amino}methyl)-6,7-dimethoxyquinolin-2-yl]piperazine-1-carboxylate
7-methoxy-4-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}quinazoline
1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}-2-phenylethane-1,2-dione
1-{4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-[5-(1H-1,3-benzodiazol-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]acetic acid
1-(2-methylphenyl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-diazepane
2-methyl-2-{4-[(1E)-pent-1-en-1-yl]phenyl}propanamide
N,N-dimethyl-2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethane-1-sulfonamide
2-[3-(1H-imidazol-1-yl)propyl]-9-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2-methyl-1-benzofuran-7-yl)-1-[(1r,4r)-4-hydroxycyclohexyl]urea
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
1-methanesulfonyl-4-[5-(5-methylfuran-2-yl)-4-phenyl-1H-imidazol-1-yl]piperidine
6-ethyl-4-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2H-chromen-2-one
2-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-2,7-diazaspiro[4.5]decan-6-one
1-[2-methoxy-5-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-{1-[1-(but-2-ynoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
4-hydroxy-1-methyl-N-[(4-methylphenyl)(thiophen-2-yl)methyl]piperidine-4-carboxamide
ethyl 1-[3-(methylsulfanyl)propyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
2-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-5-(3-methylthiophen-2-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
2-(2,4-dioxo-1,3-thiazolidin-3-yl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)acetamide
1-benzyl-8-[(2,5-dimethylphenyl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({3-methoxy-4-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]furan-2-carboxamide
(1S,5R)-N-(2-fluorophenyl)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
2-({[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)amino)ethan-1-ol
1-[(5-methylfuran-2-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
9-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1,4,9-triazaspiro[5.5]undecan-5-one
ethyl 4-[(4-{[1-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
1-(3-oxo-3-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-({3-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-1-yl}methyl)naphthalen-1-ol
N-[2-(4-ethylphenyl)ethyl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamide
1-[(3-methoxyphenyl)methyl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-6-oxopiperidine-3-carboxamide
(1S,6R)-9-[2-(morpholin-4-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
2-(1-methyl-1H-indol-3-yl)-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}acetamide
2-(2-fluoro-4-methylphenyl)-2-{methyl[2-(morpholin-4-yl)ethyl]amino}acetic acid
1-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propan-1-one
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)benzenesulfonamide
1,4-dimethyl 2-{[6-(2-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}butanedioate
5-methoxy-3-methyl-2-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-1H-indole
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[2-(3-methylphenyl)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-cyclopropanecarbonyl-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)piperidine-4-carboxamide
1-[1-(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}phenyl)ethyl]piperidine
1-(4-fluorophenyl)-3-{1-methyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}propan-1-one