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N2-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-N1-(4-methylpyridin-2-yl)ethane-1,2-diamine
4-(2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,3-thiazol-2-amine
N3-butyl-N5-cyclooctyl-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
4-{1-[3-(1H-imidazol-1-yl)propyl]-4-phenyl-1H-imidazol-5-yl}phenol
(2S,4R)-4-[(1-benzylpiperidin-4-yl)amino]-N-ethyl-1-(naphthalen-2-ylmethyl)pyrrolidine-2-carboxamide
N4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}quinolin-6-yl)acetamide
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-4-oxobutanamide
1-{2-[4-(3-benzylpyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}piperazine
(2S,4R)-N-ethyl-4-{[(4-fluorophenyl)methyl]amino}-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(pyridin-4-yl)-1,4-diazepane
2-benzyl-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-N-[2-(morpholin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(2-{4-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]phenoxy}ethyl)acetamide
4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}thiomorpholine
2-{4-[1-(3-methylbenzoyl)piperidin-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N,3,6-trimethyl-1-benzofuran-2-carboxamide
N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclobutanecarboxamide
2-[(3-{2-[methyl(2-methylpropyl)amino]ethyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)methyl]benzonitrile
4-(2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyridine-4-carbonyl)morpholine
2,6-difluoro-3-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(propan-2-yl)benzamide
2-chloro-N-{[2-(dimethylamino)pyridin-3-yl]methyl}-6-fluorobenzamide
5-{[(3-chlorophenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
9-methoxy-7-[4-(methylsulfanyl)phenyl]-4-(quinolin-6-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(oxan-4-ylmethyl)-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
2-{4-[3-(3,4-difluorophenyl)propanoyl]morpholin-3-yl}acetic acid
2-[(3-fluorophenyl)methyl]-6-methyl-3-(4-methylpiperidine-1-carbonyl)-1-[3-(morpholin-4-yl)propyl]-1,4-dihydropyridin-4-one
3-benzyl-4-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
{4-[(2-chlorophenyl)methyl]-1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-4-yl}methanol
3-{4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-3,5-dimethyl-1H-pyrazol-1-yl}propanamide
2-cyclobutanecarbonyl-5-(5-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1,2,4-oxadiazol-3-yl)-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
3-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
6-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
2-(methylamino)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1,3-thiazole-4-carboxamide
methyl 4-{2-amino-3-cyano-8-hydroxy-5H,6H-benzo[h]quinolin-4-yl}-1H-pyrazole-3-carboxylate
1-cyclopentyl-4-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
3-butyl-1-(2-{3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-oxoethyl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-1-[(5-cyclohexylthiophen-2-yl)methyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
(3S,4R)-1-[2-(4-ethylpiperazin-1-yl)acetyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]acetamide
2-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-6-(trifluoromethyl)pyridine-3-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-propyl-1H-pyrazole-5-carboxamide
1-{7-cyclopropanecarbonyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-4-ethylpiperazine
6-{1-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
1-cyclohexyl-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
[3-(1H-imidazol-1-yl)propyl]({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
3-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-(4-methylphenyl)urea
1-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)pyrrolidin-3-amine
3-sulfamoyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide