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4-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-1-ethyl-1H-pyrrole-2-carbonitrile
1-benzyl-4-({4-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[4-(quinolin-3-yl)-1H-pyrazol-1-yl]acetamide
4-[1-({5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl}amino)ethyl]hepta-1,6-dien-4-ol
3-(2,3-dihydro-1-benzofuran-7-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
4-(hydroxymethyl)-1-[(4-methanesulfonylphenyl)methyl]azepan-4-ol
4-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}morpholine
2-(dimethylamino)-1-(4-{5-[(4-hydroxypiperidin-1-yl)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
(3S,7S,8aS)-7-{[(2,5-dimethylphenyl)methyl]amino}-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-acetyl-N-(1-hydroxybutan-2-yl)-N-[(5-methylthiophen-2-yl)methyl]benzamide
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]bis(1,3-oxazol-4-ylmethyl)amine
5-methyl-3-{pyrazolo[1,5-a]pyrimidin-3-yl}-[1,2,4]triazolo[4,3-a]pyridine
4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]morpholine
1-(3-benzoylpiperidin-1-yl)-2-(2H-1,3-benzodioxol-5-yloxy)ethan-1-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
(2S,4R)-4-amino-1-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-N-methylpyrrolidine-2-carboxamide
5-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-(3-fluorophenyl)pyridine
1-methyl-4-{2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carbonyl}piperazin-2-one
3-cyclopropyl-1-(2,5-dimethylphenyl)-5-[(2-methoxyethoxy)methyl]-1H-1,2,4-triazole
2-{[4-(1,2-oxazinane-2-carbonyl)-1,3-oxazol-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
methyl (2S,4S)-1-[(2,5-dimethoxyphenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-4-(piperidin-1-ylmethyl)benzamide
4-(5-fluoro-3-methyl-1H-indole-2-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-5-methyl-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
5-[4-(pyrazin-2-yl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
8-acetyl-2-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[1-(3-methoxyphenyl)ethyl]methylamine
2-[5-(azepan-4-yl)-1-(5-chloro-2-methoxyphenyl)-1H-1,2,4-triazol-3-yl]acetamide
2-amino-6-(4-hydroxyphenyl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}({[5-(oxolan-2-yl)thiophen-2-yl]methyl})amine
1-cyclopentyl-5-[4-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propanamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[4-(2-phenoxyethyl)piperazin-1-yl]propan-1-one
5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine
5-[4-(2-ethoxyphenyl)piperazin-1-yl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
3-{1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]azetidin-3-yl}pyridine
5-{3-[2-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
N-{[5-(2-chlorophenyl)-1,2-oxazol-3-yl]methyl}-2-(furan-2-yl)-2-oxoacetamide
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(5-amino-1H-1,2,4-triazol-3-yl)propan-1-one
N-(2,6-dimethoxypyridin-3-yl)-4-[(3-oxopiperazin-1-yl)methyl]benzamide
N-(3-{4-[(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}phenyl)-3-(trifluoromethyl)benzamide
8-(quinoline-8-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
4-(5-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-2-yl}-1,2,4-oxadiazol-3-yl)pyridine
N4-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
9-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(4-{[5-(2-chlorophenyl)furan-2-yl]methyl}piperazin-1-yl)ethyl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
N-tert-butyl-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-(butan-2-yl)-N-[(2-fluorophenyl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,4-diazepan-5-one