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N-cyclobutyl-6-(4-methoxyphenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-ethyl-4-{[1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-yl]amino}pyrrolidin-2-one
2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}acetamide
4-methyl-N-[(1R,3S)-3-{[2-(pyridin-4-yl)ethyl]carbamoyl}cyclopentyl]piperazine-1-carboxamide
5-{[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N,N-dimethylpyrimidin-2-amine
1-[3-(1H-imidazol-1-yl)propanoyl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
1-(4-methanesulfonylphenyl)-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
5-(2,2-dimethylmorpholine-4-carbonyl)-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
[(3R,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)pyrrolidin-3-yl]methanol
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]acetamide
N-methyl-5-[1-(2-methylpropyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethan-1-one
2-{1-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrrolidin-2-yl}pyridine
3-(3-chlorobenzoyl)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine
2-(2,5-dimethylphenoxy)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}propanamide
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
(1S,5R)-1,3,3-trimethyl-6-(1-methyl-1H-pyrazole-4-carbonyl)-6-azabicyclo[3.2.1]octane
2-(adamantan-1-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N4-{2-[ethyl(methyl)amino]butyl}-5,6-dimethylpyrimidine-2,4-diamine
1-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(1R,4S)-2-[2-(4-ethylphenyl)pyridine-3-carbonyl]-2-azabicyclo[2.2.1]heptane
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]pyrimidine-5-carboxamide
8-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1-oxa-8-azaspiro[4.6]undecane
N-(1-{1-[2-(2-methoxyphenoxy)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)oxolane-3-carboxamide
5-methanesulfonyl-2-(4-methylpiperazin-1-yl)-4-(piperidin-3-yl)pyrimidine
(1-ethyl-5-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
N-[2-(pyridin-2-yl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
N-[3-(1,3-benzothiazol-2-yl)propyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[(4-chloro-3-fluorophenyl)methyl]-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
methyl 2-[methyl({2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})sulfamoyl]benzoate
4-({4-methyl-5-[1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
3,5-dimethoxy-2-{[(1S,6R)-3-methyl-3,9-diazabicyclo[4.2.1]nonan-9-yl]methyl}benzoic acid
3-(3-chloro-1,2-oxazol-5-yl)-1-{3,9-diazaspiro[5.5]undecan-3-yl}propan-1-one
2-benzyl-9-(2-fluoro-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-chloro-2-({3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2-methyl-1,3-benzothiazole-5-carbonyl)piperidin-3-amine
1-(4-methylphenyl)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazin-2-one
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
(2S,4S)-1-benzyl-N-(2-methoxyethyl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(1R,2R)-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-phenylcyclopropane-1-carboxamide
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}(methyl)(pyrazin-2-ylmethyl)amine
N-methyl-3-(1-methyl-1H-pyrrol-2-yl)-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-1H-pyrazole-5-carboxamide
1-[4-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
3-ethyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-4-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-(3-methoxyphenyl)-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]piperidine
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(5-cyclopropyl-1,2-oxazol-3-yl)methyl]methylamine
9-methoxy-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-fluoro-6-[1-(3-methylbutyl)-1H-pyrazol-4-yl]benzamide