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N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-4-yl)acetamide
ethyl 4-[2-(1-benzyl-3-oxopiperazin-2-yl)acetyl]piperazine-1-carboxylate
4-[4-(2,8-dimethylquinoline-3-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
(3S,4S)-4-cyclopropyl-1-{2-[3-(trifluoromethyl)phenyl]acetyl}pyrrolidine-3-carboxylic acid
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4,4,4-trifluorobutanamide
(1S)-1-[1-cyclohexyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-2-(4-methoxyphenyl)ethan-1-amine
9-methoxy-7-(6-methoxypyridin-2-yl)-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[(3-{ethyl[2-(4-fluorophenoxy)ethyl]carbamoyl}phenyl)amino]acetic acid
2-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
5-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide
N-[3-(3-fluorophenyl)phenyl]-1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidine-4-carboxamide
8-(2-methoxyethyl)-9-oxo-N-(2-phenylethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
methyl 2-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-1-oxo-1,2-dihydroisoquinoline-7-carboxylate
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]{[7-methyl-2-(morpholin-4-yl)quinolin-3-yl]methyl}amine
4-(4-ethyl-6-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyrimidin-2-yl)morpholine
4-[(3R)-3-hydroxypyrrolidine-1-carbonyl]-N-(pyridin-2-ylmethyl)benzene-1-sulfonamide
1-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
methyl 5-[(adamantan-2-yl)amino]-1-benzyl-3-cyclopropaneamido-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
3-(4-{[4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)-5-methyl-1,2,4-oxadiazole
1-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-3-{[(4-fluorophenyl)methyl]sulfanyl}propan-1-one
methyl 2-{[(4-fluorophenyl)methyl]sulfamoyl}-6-[(2E)-2-methylbut-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-2-(1H-1,2,4-triazol-5-yl)benzamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)propanamide
2-(1H-indol-1-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-amino-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
3-chloro-N-[4-(5-methylfuran-2-amido)phenyl]pyridine-4-carboxamide
1-[2-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)phenyl]ethan-1-one
N-cyclobutyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-3-methoxypropan-1-one
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[3-(morpholin-4-yl)propyl]acetamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,4-diazepan-5-one
9-(3-chloro-2-methylbenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
5-[1-(4-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(pyridin-3-yl)pyrimidine
8-cyclopropanecarbonyl-2-(furan-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(cyclopropylmethyl)-4-hydroxy-N-(2-methoxyethyl)-2-phenylpyrimidine-5-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)cyclobutanecarboxamide
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-(1,3-thiazol-2-yl)piperidine
4-(1-cyclopropanecarbonylpiperidin-4-yl)-1-(3-methoxyphenyl)-3-methylpiperazin-2-one
1-benzyl-N-ethyl-4-oxo-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
ethyl 1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidine-4-carboxylate
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4-(1-methylpiperidin-4-yl)piperazine
4-(4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-4-oxobutanoic acid
7,7-dimethyl-2-[(propane-2-sulfonyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-cyclopentyl-4-oxo-4-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butanamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-1-[(4-fluorophenyl)methyl]-N-methylpyrrolidine-2-carboxamide
2-(2-hydroxyethyl)-9-[(4-methoxy-2,5-dimethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one