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ethyl 1-methyl-5-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
[(3R,4R)-1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-cyclopentyl-5-(2-methyl-1,3-thiazole-4-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1'-(5-chloropyridin-2-yl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[4-({3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}methyl)phenyl]imidazolidin-2-one
3-({1-[1-(3-phenylpropyl)piperidin-4-yl]piperidin-4-yl}formamido)propanamide
N-[1-(5,8-dimethoxy-4-methylquinolin-2-yl)piperidin-4-yl]methanesulfonamide
2-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-3-phenoxypropan-1-one
(1S,5R)-N-(2-chloro-6-methylphenyl)-3-[(dimethylcarbamoyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
3-(2-chlorophenyl)-1-[4-(2-hydroxyethyl)piperazin-1-yl]-3-phenylpropan-1-one
N-[(3S,4R)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
4-[4-(2-methylphenyl)piperazine-1-carbonyl]-2-(1H-pyrazol-4-yl)quinoline
4-{[2-(cyclopentyloxy)phenyl]methyl}-3-(4-fluorophenyl)piperazin-2-one
6-(2-chlorophenyl)-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-4-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-[(2,3-dihydro-1,4-benzodioxin-5-yloxy)methyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole
[1-(4-aminopyrimidin-2-yl)-3-(2-phenylethyl)piperidin-3-yl]methanol
2-methoxyethyl 4-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carboxylate
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(dimethylamino)propanamide
N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}acetamide
6-{4-[(dimethylamino)methyl]phenyl}-N2,N2-dimethylpyrimidine-2,4-diamine
9-(3-ethyl-1H-pyrazole-5-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-{4-phenyl-5-[4-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}propanoate
1-{[3-(2,3-dihydro-1H-isoindole-2-carbonyl)-1H-pyrazol-5-yl]methyl}-1H-indole
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(3-chloro-5-fluorophenyl)-N,N-dimethylpyridine-3-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-[(4-phenyl-1,3-thiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-ethyl-2,3-difluoro-N-[(3R,4R)-3-hydroxy-1-(thiophene-2-carbonyl)piperidin-4-yl]benzamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
1-[2-(dimethylamino)ethyl]-4-{8-methyl-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}pyrrolidin-2-one
N-[2-(azepan-1-yl)ethyl]-N-ethyl-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
N-butyl-2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
1-(furan-2-yl)-2-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl}ethane-1,2-dione
N-(2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}ethyl)pyridine-4-carboxamide
(3aS,6aR)-5-[(4-fluorophenyl)methyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-(furan-3-ylmethyl)-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
N-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
1,3-dimethyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(1S,5R)-6-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-[3-(morpholin-4-ylmethyl)phenyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-({[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl](methyl)amino}methyl)benzonitrile
1-ethyl-4-{[2-(2-methoxyethyl)morpholin-4-yl]methyl}-1H-indole
{1-[4-(4-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
[1-(2-methylbenzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol