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{1-[2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]piperidin-3-yl}methanol
3-{1-[(5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]azetidin-3-yl}pyridine
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-(thiophene-2-carbonyl)-1,4-diazepan-2-one
3-[2-(3,4-dichlorophenyl)morpholine-4-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-(3-{[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]methyl}phenoxy)acetamide
N-(4-{[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]methyl}phenyl)acetamide
6-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]quinoxaline
N-(3-chlorophenyl)-3-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}benzamide
1-(furan-2-ylmethyl)-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidine-4-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4-[(4-phenylphenyl)methyl]piperazin-2-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[1-(4-fluorophenyl)propyl]pyrimidin-2-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-propylpiperazine
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
1-[2-({[4-(trifluoromethyl)pyridin-2-yl]amino}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]ethan-1-one
4-chloro-N,N-dimethyl-5-({methyl[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}methyl)-1,3-thiazol-2-amine
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]methylamine
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(morpholin-3-yl)acetamide
1-[2-({10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)ethyl]piperidine-3-carboxamide
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propan-1-one
(3aS,6aS)-2-(2-aminopyrimidin-4-yl)-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(1-methyl-1H-indol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-(1-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
ethyl 4-(cyclopropylmethyl)-1-[(E)-2-phenylethenesulfonyl]piperidine-4-carboxylate
(3R)-1-{5-[(diethylamino)methyl]-2-methylfuran-3-carbonyl}-3,4,4-trimethylpyrrolidin-3-ol
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carbonyl)-1,4-diazepan-5-one
2-(2,4-difluorophenoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
9-methoxy-7-oxo-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-acetyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]piperidine-3-carboxamide
3-[methyl(1-methylpyrrolidin-3-yl)amino]-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-1-one
{1-[2-({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]piperidin-2-yl}methanol
4-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-5-[3-(trifluoromethyl)phenyl]pyrimidine
2-{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-2-azaspiro[4.4]nonane
2-(3-methoxyphenyl)-N-[(3S)-2-oxoazepan-3-yl]-1,3-benzoxazole-6-carboxamide
N-cyclopropyl-5-(2,5-dihydro-1H-pyrrole-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
2-{1-[(4-methylphenyl)methyl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-2-yl}ethan-1-ol
3-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-[2-(1H-pyrazol-1-yl)phenyl]urea
(3S,4S)-4-(dimethylamino)-1-[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidin-3-ol
(4aS,8aR)-6-{[2-(ethylamino)pyrimidin-5-yl]methyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-methyl-N-{2-[5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridin-2-amine
[(3,5-dimethoxyphenyl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-{2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetyl}piperazin-2-one
1-(2-methoxyphenyl)-4-[1-(2-methylpropyl)-5-oxopyrrolidine-3-carbonyl]piperazin-2-one