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(3S,5R)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]-5-[(pyridin-2-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-(2-methoxy-4-{[(1-methylpiperidin-4-yl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-3-(3-methoxypropyl)piperidine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[2-(1H-indol-3-yl)ethyl]piperidine-3,5-dicarboxamide
3-methyl-7-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3S,9aR)-3-benzyl-8-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methoxy-5-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)benzoic acid
3-(1-butyl-1H-imidazol-2-yl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
[(3S,5R)-5-[(dimethylamino)methyl]-1-{[5-(4-methoxyphenyl)furan-2-yl]methyl}piperidin-3-yl]methanol
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
methyl[(3-phenyloxolan-3-yl)methyl]{[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
(3aS,6aS)-2-[(8-chloroquinolin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{4-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]phenyl}-N-methylmethanesulfonamide
4-(3-benzyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperazine-1-carbaldehyde
4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
3-amino-1-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
2-methyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-4,5,6,7-tetrahydro-2H-indazole
7-ethyl-2-(5-methyl-2H-1,2,3-triazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(diethylamino)-3-[2-methoxy-5-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
5-{5-[2-(furan-2-yl)-2-phenylethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[(3R,4S)-4-cyclopropyl-1-[2-(phenylsulfanyl)acetyl]pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
5-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-5-(2-methylpropyl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
N-[3-(cyclohexylcarbamoyl)-2-methylphenyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
2-(2-{1-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-N-cyclopentylpiperidine-1-carboxamide
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
3-(3,4-dimethoxyphenyl)-1-[3-(phenylamino)piperidin-1-yl]propan-1-one
5-methyl-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]-1,2-oxazole-4-carboxamide
1-(4-{[methyl(oxan-4-yl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
(3S,4S)-1-[(2-methoxypyrimidin-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
5-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[5-(2,3-dimethoxy-5-methylphenyl)-1H-1,3-benzodiazol-2-yl]methanol
N-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
3-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-3H,4H-pyrido[3,2-d]pyrimidin-4-one
4-[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]-1-(2-phenylethyl)piperazin-2-one
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-N,N-dimethylacetamide
{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}(methyl)[(3-methyl-1H-indol-2-yl)methyl]amine
1-[(2,6-difluorophenyl)methyl]-3-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
5-butyl-1'-(1-methyl-1H-pyrrole-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
1-(2,3-dihydro-1H-inden-2-yl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-5-methyl-4-(thiophen-2-yl)pyrimidine
2-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,4-diazepan-6-yl}acetic acid
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-{[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}propanamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-({4-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)acetic acid
(2R,3R,6R)-5-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[2-(dimethylamino)-4-{[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-(5-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazol-3-yl)pyridine
4-[4-(cyclopentylmethyl)-2-oxopiperazin-1-yl]benzonitrile