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methyl N-({1-[(3S,5S)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazol-4-yl}methyl)-N-methylcarbamate
3-(azepane-1-carbonyl)-1-ethyl-N-[2-methyl-2-(morpholin-4-yl)propyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-methyl-2-phenyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]furan-3-carboxamide
3-[1-(2-cyclohexylacetyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
5-(4-chlorophenyl)-N-[(1-methylpiperidin-2-yl)methyl]-1,2,4-triazin-3-amine
2-(dimethylamino)-2-(3-methylphenyl)-N-[3-(methylsulfanyl)propyl]acetamide
4-{5-[2-(methylsulfanyl)ethyl]-3-phenyl-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
9-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(methylsulfanyl)-N-[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]acetamide
(3R,4S)-4-[({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)(methyl)amino]oxolan-3-ol
5-amino-4-chloro-N-{[(1r,4r)-4-(methylcarbamoyl)cyclohexyl]methyl}-1H-pyrazole-3-carboxamide
N-[2-(4-chlorophenyl)ethyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
4-[6-oxo-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-1H-pyrazole-3-carboxylic acid
2-{4-benzyl-1-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-2-[(2-methylphenyl)sulfanyl]acetamide
4-(1-butyl-1H-imidazol-2-yl)-1-(3-chlorothiophene-2-carbonyl)piperidine
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
2-{2-[4-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,3-benzodiazole
2-{2-[1-(4-cyclopentylpyrimidin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
6-methyl-N-[(3-methylpyridin-2-yl)methyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-4-oxo-3,4-dihydroquinazoline-2-carboxamide
5-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
N-(1-methyl-1H-indazol-3-yl)-2-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-1-yl]acetamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-ethyl-N-methyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-(naphthalen-1-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4S)-1-(3-chloro-2-fluorobenzoyl)-3,3,4-trimethylpiperidin-4-ol
(3ar,6ar)-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(dimethylamino)-2-(3-methylphenyl)-1-[4-(pyridin-4-yl)piperazin-1-yl]ethan-1-one
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(furan-2-ylmethyl)-1H-pyrazole-4-carboxamide
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-fluoropiperidine-1-carboxamide
3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-1-[4-(3-methylpiperidine-1-carbonyl)phenyl]urea
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
7-(4-methylpiperidine-4-carbonyl)-N4-(propan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
7-(1,3-benzothiazol-2-yl)-4-(4-methoxybenzoyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]pyridine-3-carboxylic acid
8-(3-methoxypropyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
5,7-dimethyl-N-(oxolan-2-ylmethyl)-N-({3-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
N'-(2-{1-[(3-fluoro-2,4-dimethylphenyl)methyl]piperidin-3-yl}ethyl)ethanediamide
{1-[(3-ethenylphenyl)methyl]-3-(prop-2-en-1-yl)piperidin-3-yl}methanol
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}bis(1,3-oxazol-4-ylmethyl)amine
methyl 3-[(3S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
1-[1-benzyl-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
(1R,2S)-1-{2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}-2,3-dihydro-1H-inden-2-ol
1-(4-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenyl)imidazolidin-2-one
N,N-diethyl-4-{[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}aniline
N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-{3-methyl-5-[(3-phenylpyrrolidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl}pyridine
8-(4,6-dimethylpyrimidin-2-yl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-(2-methoxyacetyl)-N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)piperidine-3-carboxamide