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1-(1-cyclohexanecarbonylpiperidin-4-yl)-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-methyl-3-{2-oxo-2-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
4-[4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperazin-1-yl]quinazoline
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
8-(but-3-en-1-yl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
4-[2-chloro-4-(piperidine-1-carbonyl)phenoxy]-1-methanesulfonylpiperidine
2-{5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}acetic acid
4-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl]phenol
(2S,3S)-2-({[4-(2-methoxyphenyl)phenyl]carbamoyl}amino)-3-methylpentanamide
4-(5-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
(2S,4R)-N-ethyl-4-(2-hydroxyacetamido)-1-(3-methoxy-5-methylthiophene-2-carbonyl)pyrrolidine-2-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-1-methyl-1H-pyrazole-5-carboxamide
1-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-3-(5-methyl-1,3,4-thiadiazol-2-yl)urea
2-(cyclopropylmethyl)-8-(2-methoxy-3-methylbenzoyl)-2,8-diazaspiro[5.5]undecan-3-one
[(3R,4R)-4-(pyrrolidin-1-ylmethyl)-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-yl]methanol
1-({2-[3-(azocan-1-yl)-2-hydroxypropoxy]-4-methoxyphenyl}methyl)azetidin-3-ol
2,5-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]furan-3-carboxamide
N-[2-(4-fluorophenyl)-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
(2S,4S)-1-{[4-(benzyloxy)phenyl]methyl}-N-[2-(2-methoxyphenyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
5-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
{[2-(butan-2-yloxy)-3-methoxyphenyl]methyl}[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]methylamine
1-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
3-(1,5-dimethyl-1H-pyrazol-4-yl)-1-[1-(thian-4-yl)piperidin-4-yl]urea
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-{[3-(trifluoromethoxy)phenyl]methyl}urea
2-{1-[5-(3-chlorophenyl)-1,2,4-triazin-3-yl]piperidin-4-yl}-5-fluoro-1H-1,3-benzodiazole
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[(2R,3R)-1'-(1-benzofuran-2-ylmethyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
3-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-pyrazol-5-amine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl 4-{[3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamido]methyl}benzoate
(3aS,6aS)-5-(1-methylpiperidin-4-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(2-{4-[3-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)morpholine
2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]acetamide
N-(cyclohex-1-en-1-ylmethyl)-2-(1H-imidazol-2-yl)benzamide
2-amino-4-(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)-6-(6-methoxypyridin-3-yl)pyridine-3-carbonitrile
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidine-4-carboxylic acid
5-butyl-1'-(4,6-dimethylpyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3R,4R)-1-(5-fluoropyrimidin-2-yl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
methyl 3-(2-methoxyacetamido)-5-[(naphthalen-2-ylformamido)methyl]benzoate
7-[2-(adamantan-1-ylsulfanyl)acetyl]-2-amino-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(2,4-difluorophenyl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
6-methoxy-1-methyl-2-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-indole
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(trifluoromethyl)phenyl]urea
4-{4-[(2,6-difluoro-3-methoxyphenyl)methyl]piperazin-1-yl}benzoic acid
3-(1-tert-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)pyridin-2-ol
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxylic acid
5-(2-fluorophenyl)-N-[1-(pyrimidin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{[(3R,4R)-1-[5-chloro-3-(trifluoromethyl)pyridin-2-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[3-(4-fluorophenyl)-1H-indazol-1-yl]acetamide