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N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(2-oxopyrrolidin-1-yl)benzamide
4-(5-aminopyridin-2-yl)-N,N-diethylbenzamide
1-(3-{3-[1-(2-methoxyethyl)-1H-pyrazol-3-yl]phenyl}phenyl)ethan-1-one
1-{2-[5-(piperidine-1-carbonyl)thiophen-2-yl]pyrrolidin-1-yl}-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-benzyl-1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-ethylpiperidine-4-carboxamide
(2R,3R)-3-{methyl[3-(pyrrolidin-1-yl)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-(cyclobutylamino)-1-cycloheptylpyrrolidin-2-one
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[2-(2,3-dimethoxyphenyl)ethyl]pyridin-2-amine
(2S,4R)-4-amino-1-[(2-hydroxy-4-methylquinolin-6-yl)sulfonyl]-N-methylpyrrolidine-2-carboxamide
3-(4,5-dimethyl-1H-1,3-benzodiazol-6-yl)-1-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]urea
1-(3,4-difluoro-5-hydroxyphenyl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxylic acid
2-(1-methyl-1H-imidazol-2-yl)-1-[3-(oxolan-3-yl)propyl]-1H-imidazole
4-methyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
6-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-5-(trifluoromethyl)pyridine
(3aS,6aS)-2-(2-methylpropyl)-5-[2-(methylsulfanyl)pyridine-3-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(cyclohex-1-en-1-yl)-1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-N-(pyridin-2-ylmethyl)cyclopropanamine
6-methyl-1-[2-(methylsulfanyl)phenyl]-4-[(2,4,5-trimethoxyphenyl)methyl]piperazin-2-one
5-acetyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}thiophene-2-carboxamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
methyl 3-cyclobutaneamido-5-{[(2,3-difluorophenyl)methyl]amino}-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(4-{2-[(2-methylphenyl)carbamoyl]acetyl}morpholin-3-yl)acetic acid
(3S,5R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxylic acid
6-[(2-fluorophenyl)methoxy]-1-[(4-methoxyphenyl)methyl]-4-(1H-pyrazol-3-ylmethyl)-1,4-diazepan-2-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
5-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-2,2-dimethylthiomorpholin-3-one
3,6-dimethyl-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}pyrazin-2-amine
1-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
N-cyclopropyl-1-(2-methoxyphenyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
3-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}benzonitrile
3-{[(4-ethoxyphenyl)methyl]amino}-N-[(1S)-1-phenylethyl]-5-[(propan-2-yl)sulfamoyl]benzamide
3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]-4-(thiophen-2-ylmethyl)piperazin-2-one
1-amino-N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}cyclopropane-1-carboxamide
1-[(4-fluorophenyl)methyl]-4-(6-methylpyridine-3-carbonyl)-2-(propan-2-yl)-1,4-diazepane
N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{1-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)isoquinoline
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
(1R,5R)-N,N-dimethyl-6-(4-methyl-1,3-thiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
5-[(1-benzylpiperidin-4-yl)amino]-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-hydroxy-3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
6-[2-(aminomethyl)-4-fluoro-2,3-dihydro-1-benzofuran-7-yl]-N,N-dimethylpyrazine-2-carboxamide
7-{[4-(propan-2-yl)phenyl]methyl}-2-[2-(1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
(3R,4R)-1-(2,3-difluoro-4-methoxybenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
(1S,5R)-3-[2-(4-fluoro-3-methylphenyl)acetyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methyl-1-{7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)methanesulfonamide
1'-({2,4-dimethyl-5H,6H-furo[2,3-d]pyrimidin-6-yl}methyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one