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1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}-4-methylpiperazine
{2-[1-(2,4-dimethoxybenzenesulfonyl)piperidin-2-yl]ethyl}dimethylamine
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
5-{[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
4-ethyl-6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-[(4-methoxyphenyl)methyl]piperazin-2-one
N-{2-[(pyridin-3-yl)amino]ethyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-[(2S,4R,6R)-2-benzyl-6-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]oxan-4-yl]acetamide
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2-methyl-4-phenylpyridine-3-carboxamide
2-benzyl-4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)morpholine
2-(1-{[1-(3,3-dimethylbutyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
5-(2-fluorophenyl)-2-(pyridin-3-yl)-4-[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]pyrimidine
1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]cyclopropane-1-carboxamide
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-methyl-1H-pyrazol-1-yl]-5-methyl-4-(thiophen-2-yl)pyrimidine
[3-({1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
2-(1-{1-[(3-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl}propyl)-2,3-dihydro-1H-isoindol-1-one
4-methyl-5-[4-(piperidine-1-carbonyl)piperidine-1-carbonyl]pyrimidine
1-(3-fluorophenyl)-3-{1-[1-(pyridine-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-(5-fluoro-2-methoxyphenyl)-1,3-benzothiazole
N-{4-[2-(2-hydroxyethyl)-4-methyl-1H-1,3-benzodiazol-1-yl]phenyl}acetamide
4-hydroxy-2-({3-[(methylsulfanyl)methyl]piperidin-1-yl}methyl)quinoline-6-carboxamide
4-{4-[(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)methyl]phenyl}-2-methylbut-3-yn-2-ol
4-({1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)-1,5-dimethyl-1H-pyrrole-2-carbonitrile
methyl({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)(quinolin-5-ylmethyl)amine
(2S,4R)-1-(1-methylpiperidin-4-yl)-N-(propan-2-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
1-[3-(morpholin-4-yl)propyl]-5-(4-phenylpiperazine-1-carbonyl)piperidin-2-one
1-{2-[(3-chlorophenyl)methyl]-1,3-benzoxazole-6-carbonyl}piperidin-4-ol
2-(4-methyl-6-{4-[methyl(1,2-oxazol-3-ylmethyl)amino]piperidin-1-yl}pyrimidin-2-yl)phenol
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
3,5-dimethyl-4-({2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-1,2-oxazole
(4aS,7aR)-1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3-{[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)carbamoyl]amino}phenyl)cyclopentanecarboxamide
N-methyl-4-oxo-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-[1-(propan-2-yl)piperidin-4-yl]-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}acetamide
4-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-2-phenylpiperazine
N-({5-[(3-fluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-phenyl-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
8-(butan-2-yl)-1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{4-benzyl-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-yl}methanol
1-{[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-{2-[3-(4-tert-butylphenoxymethyl)-1-ethyl-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-4-(3-methylphenoxy)piperidine-4-carboxylic acid
1-[(1-{6-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-benzyl-1-(1-methyl-1H-indole-6-carbonyl)piperidin-4-ol
2-methoxy-6-({methyl[(3-methyl-1H-indol-2-yl)methyl]amino}methyl)phenol