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1-(3-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-{1-[(3-chlorophenyl)methyl]piperidin-4-yl}-5-ethylimidazolidine-2,4-dione
2-(4-methylphenyl)-1-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
3-({[(tert-butylcarbamoyl)methyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-{[2-(dimethylamino)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]-4-methylbenzamide
1-cyclopentyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
dimethyl[(2-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]methyl}phenyl)methyl]amine
2-{4-[1-(4-fluoro-2-methylphenyl)piperidin-4-yl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
[(3R,4R)-1-[(3,5-difluorophenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
3-(2-fluorophenyl)-5-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
methyl (1R,3S,3aR,6aS)-3-(2-aminopyrimidin-5-yl)-5-ethyl-1-(2-methylpropyl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
(3R,5R)-N-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
[3-(hydroxymethyl)-4-[4-(1H-pyrazol-5-yl)phenyl]phenyl]methanol
3-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
5-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyridine-3-carboxamide
1-(2,2-diphenylethyl)-5-{2-[(2-methoxyethyl)amino]ethyl}pyrrolidin-2-one
2-{[2-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
3-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-9-methyl-3,9-diazaspiro[5.6]dodecane
2-[7-chloro-2-(furan-2-yl)-8-methylquinoline-4-carbonyl]-1,2-oxazolidin-4-ol
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
2-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}acetic acid
3-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-N-(1,2,3-thiadiazol-5-yl)benzamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
methyl 4-(2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)butanoate
ethyl 5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-[3-(benzyloxy)phenyl]-3-cyanopiperidine-1-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-4,6-dimethyl-2-oxo-N-propyl-1,2-dihydropyridine-3-carboxamide
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(pyridin-3-yl)ethan-1-one
4-[1-(4-chloro-2,5-dimethylbenzenesulfonyl)piperidin-3-yl]morpholine
2-(2,4-dimethoxyphenyl)-5-methyl-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1,3-oxazole
N-{[3-(difluoromethoxy)phenyl]methyl}-4-(piperidin-3-yl)benzamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-{4-[6-methyl-2-(methylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
3-[1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
N-(3-methylphenyl)-3-[2-(4-propanoylphenoxy)acetamido]propanamide
3-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-1-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}urea
3,5-dichloro-4-methyl-N-(1,4-oxazepan-6-ylmethyl)benzamide
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
(3R,4S)-4-(4-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,4-diazepan-1-yl)oxolan-3-ol
N-(3-chloro-4-fluorophenyl)-3-[1-(2-methyl-1H-pyrrole-3-carbonyl)piperidin-4-yl]propanamide
4-ethyl-3-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)benzonitrile
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-[4-(4-fluorophenyl)piperazin-1-yl]propan-1-one
4-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
3-[(3-chlorophenyl)methyl]-N-[2-(methylsulfanyl)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl][2-(1H-imidazol-1-yl)ethyl]methylamine