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(3R,4S)-1-[(dimethyl-4H-1,2,4-triazol-3-yl)methyl]-3,4-dimethylpiperidin-4-ol
2-{[(4-fluorophenyl)methyl]({[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl})amino}butan-1-ol
4-hydroxy-N-[(1S,2S)-2-hydroxycyclohexyl]-2-phenylpyrimidine-5-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(furan-2-yl)azepane
7-[(2,3-difluorophenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decane
(3aR,6aR)-2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(1S,5R)-6-(propane-1-sulfonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2-{1-[4-(3-methoxyphenyl)benzoyl]piperidin-2-yl}ethyl)dimethylamine
8-[1-(methoxymethyl)cyclopropanecarbonyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-amino-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)cyclopropane-1-carboxamide
2-ethyl-4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
[3-(cyclopropylmethyl)-1-(2-methylpyrimidine-5-carbonyl)piperidin-3-yl]methanol
4-{[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amino}-1λ4-thian-1-one
1-(2-methylphenyl)-3-(2-methylpropyl)-5-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
N-cyclopropyl-N-({4-[(2,5-dimethoxyphenyl)methoxy]phenyl}methyl)-2H-1,3-benzodioxole-5-carboxamide
3-(2-ethylbutyl)-8-[2-(pyridin-4-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-ethyl-3,5-dimethyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1H-pyrazole-4-carboxamide
N-(2-fluoro-4-methylphenyl)-3-(3-methoxypropyl)piperidine-1-carboxamide
1-(cyclopropylmethyl)-5-(4-methylpyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-({methyl[3-(5-methylfuran-2-yl)butyl]amino}methyl)-3,4-dihydroquinazolin-4-one
2-tert-butyl-7,7-dimethyl-N-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydroquinazolin-5-amine
[(2,4-difluorophenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
2-(1H-imidazol-1-yl)-1-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)ethan-1-one
6-propyl-2-(4-{[4-(pyrrolidin-1-yl)piperidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-1-(3,4,5-trimethoxyphenyl)urea
6-fluoro-2-{[3-(2-methoxybenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
N-[2-(2-ethylphenoxy)ethyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
methyl 6-(azepan-1-ylmethyl)-3-(furan-2-amido)thieno[2,3-b]pyridine-2-carboxylate
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]imidazo[1,2-a]pyrimidine-2-carboxamide
4-({[1-(2-methoxyphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)pyridine
2-(4-fluorophenyl)-1-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
5-(2-chlorophenyl)-N-[(3-methyloxetan-3-yl)methyl]furan-2-carboxamide
4,6-dimethyl-2-oxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N4-[(2-ethoxypyridin-3-yl)methyl]-5-ethylpyrimidine-2,4-diamine
1-benzyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2-ethoxypyridin-3-yl)methyl]-N'-(2,4,6-trimethylphenyl)butanediamide
3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]-1-(2-phenylpropyl)piperidine
methyl 6-[(5-chloro-2-hydroxyphenyl)methyl]-2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidin-4-ol
1-cycloheptyl-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
ethyl 1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-(2-phenylethyl)piperidine-3-carboxylate
N-[2-(7-fluoro-2-methylquinoline-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
3-(pyrrolidin-3-yl)-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
2-[4-(methylsulfanyl)phenyl]-3-(pyrrolidin-1-yl)pyrazine
2-chloro-4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]phenol
2-(2-methoxyphenyl)-N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]acetamide
3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
5-[2-(dimethylamino)propanoyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-{3-cyclopentyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-(oxan-2-ylmethoxy)ethan-1-one