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N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamide
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
5-{[(3-methoxyphenyl)methyl]amino}-N,N-dimethyl-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-[({2-[2-hydroxy-3-(4-hydroxypiperidin-1-yl)propoxy]-5-methoxyphenyl}methyl)(methyl)amino]-N-methylacetamide
3-fluoro-N-{1-[1-(3-fluoropyridin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
N-butyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)acetamide
1-(dimethyl-1,2-oxazol-4-yl)-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
(3R,4R)-4-cyclobutyl-3-methyl-1-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-ol
9-(3-methoxypyrazin-2-yl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
4-(hydroxymethyl)-1-{2-[(2-methoxyethyl)amino]-1-methyl-1H-1,3-benzodiazole-5-carbonyl}piperidin-4-ol
(3S,5S)-5-[(6-methylpyridin-3-yl)carbamoyl]-1-(2-phenylethyl)piperidine-3-carboxylic acid
1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-[2-(methylsulfanyl)benzoyl]piperidine
N-(3-fluorophenyl)-3-[4-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
5-(4-phenoxyphenoxy)-1-azabicyclo[3.2.1]octane
(1,3-benzoxazol-2-ylmethyl)({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
1-(methoxymethyl)-N-[(4-sulfamoylphenyl)methyl]cyclobutane-1-carboxamide
{2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
1-[(4-fluorophenyl)methyl]-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-2-one
1-(3-{4-[(4-fluoropiperidin-1-yl)methyl]-2-methoxyphenoxy}-2-hydroxypropyl)piperidin-4-ol
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(1-methyl-1H-indazol-6-yl)urea
3-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]propanamide
3-(1H-indazol-5-yl)-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
(2E)-2-methyl-N-{[7-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}but-2-enamide
2,4-dimethyl-N-[1-(4-{[(5-phenyl-4H-1,2,4-triazol-3-yl)methyl]carbamoyl}phenyl)-1H-pyrazol-4-yl]benzamide
4-{[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
N-benzyl-5-[(3-ethoxyphenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aS,6aS)-2-{5-[(dimethylamino)methyl]furan-2-carbonyl}-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{2-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]phenyl}-1H-1,2,4-triazole
[2-(1H-imidazol-1-yl)ethyl](methyl){[5-(oxolan-2-yl)thiophen-2-yl]methyl}amine
[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]methanamine
2-[5-(1-cyclopentanecarbonylpiperidin-4-yl)-3-phenyl-1H-1,2,4-triazol-1-yl]ethan-1-ol
(4aR,7aS)-1-methanesulfonyl-4-(3-phenylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-1-(2H-1,3-benzodioxol-5-ylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
3-{2-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
6-cyclopentyl-2-methoxy-3-{[(pyrimidin-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(4-methoxyphenyl)-3-methyl-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperazin-2-one
N-cyclooctyl-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
1-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)ethan-1-one
1-cyclohexyl-4-(5-methyl-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)piperazine
1-(2-methyl-1-benzofuran-7-carbonyl)-3-(1-methyl-1H-imidazol-2-yl)piperidine
(2S,4R)-1-(1H-indol-5-ylmethyl)-N-methyl-4-[3-(methylsulfanyl)propanamido]pyrrolidine-2-carboxamide
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-(2,4,5-trimethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(3-chlorophenyl)methyl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
3-{methyl[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propanamide