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2-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-3-methylquinoxaline
1,3,6-trimethyl-N-[1-(pyrazin-2-yl)propan-2-yl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[2-(ethylamino)pyrimidin-5-yl]-N,N,6,8-tetramethylquinoline-4-carboxamide
ethyl 1-(3-{[2-(1-methylpyrrolidin-2-yl)ethyl]carbamoyl}-6-(4-methylthiophen-2-yl)pyridin-2-yl)piperidine-4-carboxylate
4-cyclobutanecarbonyl-9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 1-{[4-(5-chloro-2-fluorobenzoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-4-carboxylate
N-[2-(N-methylmethanesulfonamido)ethyl]-4-(piperidin-3-yl)benzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-N-{[6-(morpholin-4-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}cyclobutanecarboxamide
1-methyl-4-(4-methylpent-3-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2,5-difluoro-N-(1-{7-[(4-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
1,3-dimethyl-5-{[(9H-purin-6-yl)amino]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N4,N4-diethyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine-2,4-diamine
3-(azocan-1-yl)-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]propanamide
1-(furan-2-ylmethyl)-N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)piperidine-4-carboxamide
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-[(2-methylphenyl)methyl]piperazine
5-[2-(methylsulfanyl)phenoxymethyl]-3-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrole-1-carbonyl]-1,2-oxazole
N-cyclopropyl-2-phenyl-N-(thiophen-3-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
(2S,4R)-1-(2-methylpropyl)-N-(propan-2-yl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-[2-(3,4,5-trifluorophenyl)acetyl]pyrrolidine-3-carboxylic acid
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
5,7-dimethyl-N-{3-[(1-methylpiperidin-4-yl)oxy]propyl}pyrido[2,3-d]pyrimidin-4-amine
2-(4-methoxyphenoxymethyl)-N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1,3-oxazole-4-carboxamide
2-{[5-(1,2-oxazol-5-yl)thiophen-2-yl]sulfonyl}-2,8-diazaspiro[4.5]decane
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-4-(pyridin-3-yl)pyrimidin-2-amine
N-{2-[(1-benzoylpiperidin-4-yl)amino]ethyl}-2,2,2-trifluoroacetamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanamide
N-[2-(2-hydroxyethoxy)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-phenylpiperidin-4-ol
3-[(3-fluorophenyl)methyl]-5-(pyrrolidin-1-ylmethyl)-1,2,4-oxadiazole
3-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-[2-(methylsulfanyl)phenyl]urea
5-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1-(2-phenylethyl)piperidin-2-one
4-methyl-2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
N-cyclopropyl-N-{[2-(4-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2,2-diphenylacetamide
1-(4-{5-[3-(diethylamino)pyrrolidine-1-carbonyl]-2-methoxyphenoxy}piperidin-1-yl)ethan-1-one
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1,2,3,4-tetrahydroquinoline-8-carboxamide
N,5-dibenzyl-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(phenylamino)-1-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]butan-1-one
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-5-(morpholine-4-carbonyl)pyridin-2-amine
3-methyl-1-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazol-5-amine
7-(4-methoxy-2-methylbenzoyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-(3-methoxypropyl)-8-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
[1-(2H-1,3-benzodioxole-5-carbonyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
1-{6-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
4-ethyl-5-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-N-[1-(thiophen-3-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
(1S,4S)-2-[(1-{[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]-2-azabicyclo[2.2.1]heptane
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(2S,4S)-4-(4-{[1-(2-chloro-5-fluorophenyl)-N-methylformamido]methyl}-1H-1,2,3-triazol-1-yl)-N-methylpyrrolidine-2-carboxamide
5-[2-(2,3,6-trimethylphenoxy)acetyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid