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N-ethyl-2-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidin-4-amine
N-[1-(methoxymethyl)cyclopentyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
4-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-1,4-oxazepane
N-tert-butyl-2-{[4-(ethylamino)pyrimidin-2-yl]amino}acetamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[4-(3-fluorophenyl)phenyl]-3-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]urea
1-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-2-(4-methoxyphenyl)acetamide
4-{1-benzyl-5-[(2,6-difluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperazin-2-one
8-[2-(morpholin-4-yl)-2-oxoethyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
8-(2-methyl-4-phenyl-1,3-thiazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-(1-{1-[(3-chloro-4-fluorophenyl)methyl]piperidin-4-yl}ethyl)morpholine
N-[1-(4-chlorophenyl)ethyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4'-ethyl-3'-oxo-N-(prop-2-en-1-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-carboxamide
N-cyclopentyl-5-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-1H-pyrazole-3-carboxamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[2-(N-methylmethanesulfonamido)ethyl]acetamide
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)quinoxaline-5-carboxamide
3-(2-fluorophenyl)-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
(3aS,6aS)-5-{3-carbamoyl-5H,6H,7H-cyclopenta[b]pyridin-2-yl}-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-phenylpiperazin-1-yl)-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]propan-1-one
4-(3-hydroxy-3-methylbutyl)-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]benzamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(3-cyano-2-methyl-1H-indol-1-yl)acetamide
(3S,5R)-N3-cyclohexyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
5-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-1,3-oxazole-4-carboxamide
1-(1-benzothiophen-2-ylmethyl)-4-(1H-pyrrole-2-carbonyl)piperazine
1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
(5S,9aS,9bS)-2-[(4-methoxyphenyl)methyl]-5-[1-(pyridin-3-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-(3-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-(4-phenyl-1H-pyrazol-5-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
(3S,4S)-1-(2,1,3-benzothiadiazol-4-ylmethyl)-4-(3-methoxyphenyl)piperidin-3-ol
1-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-3-ylmethyl)-1,4-diazepane
3-(1-methyl-1H-pyrazol-4-yl)-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]propanamide
3-(5-{[4-(pyridin-3-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
[5-(6-chloro-1H-1,3-benzodiazol-2-yl)-2-ethoxyphenyl]methanol
[1-(2,6-dimethylpyridine-4-carbonyl)piperidin-4-yl](thiophen-2-yl)methanol
(3S,4R)-1-(2,3-difluoro-6-methoxybenzoyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
1-methyl-5-{[3-(propan-2-yloxy)propyl]amino}-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(2,3-difluoro-6-methoxybenzoyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
N,N-dimethyl-5-[methyl(thiophen-2-ylmethyl)amino]-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-3-(1-methylpiperidin-3-yl)propan-1-one
3-{3-[(2-methoxyphenyl)methyl]-1-(6-methylpyridin-2-yl)-1H-1,2,4-triazol-5-yl}propanamide
6-[4-(2-methoxyethyl)piperazine-1-carbonyl]-N-[2-(3-methoxyphenyl)ethyl]-5-methylthieno[2,3-d]pyrimidin-4-amine
(2S,4R)-N-ethyl-4-(3-hydroxypropanamido)-1-[2-(4-methylphenyl)acetyl]pyrrolidine-2-carboxamide
5-{1-[5-(ethylsulfanyl)thiophene-2-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-ethyl-5-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}piperidin-2-one
3-(2,5-dimethylphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
N-[(4-fluorophenyl)methyl]-6-oxo-N-(oxolan-2-ylmethyl)-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(2-methoxy-4-methylphenoxymethyl)-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
2-(2-aminoethyl)-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylquinazolin-4-amine