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5-{4-[2-(5-fluoro-2-methyl-1H-indol-3-yl)acetyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
1-[4-(1H-imidazol-1-yl)benzoyl]-3-[(methylsulfanyl)methyl]piperidine
6-oxo-1-(3-phenylpropyl)-N-[2-(pyridin-4-yl)ethyl]piperidine-3-carboxamide
N-[(2S)-1-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-4-(methylsulfanyl)-1-oxobutan-2-yl]acetamide
N-[(2S)-1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-4-methyl-1-oxopentan-2-yl]acetamide
methyl 6-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}pyrazine-2-carboxylate
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
1-[4-({cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
2-{[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]methyl}benzonitrile
(3S,4R)-1-(3-methylfuran-2-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
2-cyano-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}benzamide
N-methyl-3-[2-({[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]carbamoyl}amino)phenyl]propanamide
2-ethoxy-5-{1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}pyridine
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-N-(pyridin-3-ylmethyl)-2-(trifluoromethyl)benzamide
6-(2-methoxyphenyl)-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[4-(azepan-1-ylmethyl)phenyl]-6-butyl-3,4-dihydropyrimidin-4-one
2-[4-(3-chlorophenyl)-2-methyl-5-oxopiperazine-1-carbonyl]benzonitrile
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-methyl-N-(oxolan-2-ylmethyl)-1,3-thiazole-4-carboxamide
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]ethan-1-one
2-(3-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenoxy)acetic acid
(1S,5R)-3-[(dimethylcarbamoyl)methyl]-N-[2-(methylsulfanyl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
5-(4-chlorophenyl)-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-1,2,4-triazin-3-amine
N-ethyl-N-[(2E)-3-phenylprop-2-en-1-yl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
4-[3-(2-fluorophenyl)propanoyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2,6-dimethyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}quinoline-3-carboxamide
3-(1-{3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl}piperidin-3-yl)propan-1-ol
1-(cyclohexylmethyl)-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
(benzylsulfamoyl)({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl})amine
4-(3-fluorophenoxy)-1-[1-(2-methoxyethyl)piperidine-4-carbonyl]piperidine
[4-({[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl](methyl)amino}methyl)oxan-4-yl]methanol
1-{4-[1-(4-fluoro-3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-4-oxobutyl}pyrrolidin-2-one
N-(1-ethyl-5-oxopyrrolidin-3-yl)-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[3-(5-methyl-1,2,4-oxadiazol-3-yl)benzoyl]pyrrolidine-2-carboxamide
1-(3,5-difluorophenyl)-N-(oxan-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[(3,4-dichlorophenyl)methyl]-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-(1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}azetidin-3-yl)pyridine
1-[2-(benzyloxy)ethyl]-3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
4-(2-benzyl-1,3-thiazole-4-carbonyl)thiomorpholine
2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}-1,3-thiazole
3,5-dimethyl-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2-oxazole-4-carboxamide
(4S)-3-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
2-[4-(propan-2-yl)phenyl]-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
1-ethyl-4-({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)piperazine
(1R,5R)-N,N-dimethyl-6-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
6-methyl-5-{1H-pyrazolo[3,4-b]pyridin-1-yl}pyridin-2-amine
2-(3-methoxypropyl)-8-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-(2-methylphenyl)-N-[2-(1-methylpiperidin-3-yl)ethyl]propanamide
1-(5-propyl-1,2-oxazole-4-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine