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2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
1-(6-methyl-2-propylpyrimidin-4-yl)-N-(pyridin-4-ylmethyl)piperidin-4-amine
N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-[2-(pyrrolidin-1-yl)ethyl]piperidine-3-carboxamide
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-cyclopropylacetamide
6-(cyclopropylamino)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]pyridine-3-carboxamide
(2E)-3-(3-fluorophenyl)-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]prop-2-enamide
[1-(1,4-dioxane-2-carbonyl)piperidin-4-yl]diphenylmethanol
1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
N-[(1R,3R)-3-aminocyclopentyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
{5-methyl-7-[2-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
(3R,7S,8aS)-3-(hydroxymethyl)-7-{[(3-methylphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
1-(cyclopropylmethyl)-6-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-3-(isoquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]-N-[4-(2-hydroxyethyl)phenyl]benzamide
(3R,5S)-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyrrolidin-3-amine
6-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-N,N-dimethylpyrazine-2-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(propan-2-yl)pyrimidine-4-carboxamide
1-(2-cyclopropylquinoline-4-carbonyl)-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
2-[9-(2-hydroxy-4-methylbenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
[(3-ethenylphenyl)methyl](methyl)[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amine
4-{[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]sulfamoyl}-N-(propan-2-yl)benzamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[(4-methylphenyl)methyl]propanamide
3-[(cycloheptylamino)methyl]-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-2-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}propanamide
N,1,3-trimethyl-N-[2-(oxan-2-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[4-(1-{[1-(methoxymethyl)cyclopropyl]methyl}-1H-imidazol-2-yl)phenyl]pyridine
N-(3-methoxypropyl)-2-(3-methyl-1H-pyrazol-1-yl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}acetamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(3-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-ethyl-N-(oxan-4-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(2R,3R)-3-({[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]acetamide
N-(2,4-dimethoxyphenyl)-3-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]propanamide
N-({1-[(3-ethyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}methyl)-2H-1,3-benzodioxole-5-carboxamide
4-benzyl-3-ethyl-1-(pyridin-2-ylmethyl)-1,4-diazepan-5-one
5-(2-ethylphenyl)pyridine-2-carbonitrile
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1,3-benzothiazole
N-benzyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-1-(4-methoxyphenyl)piperidine
(4S)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-[3-(1H-imidazol-5-yl)phenyl]-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
1-(3-methylbut-2-en-1-yl)-3-[2-(methylsulfanyl)benzoyl]piperidine
(2S,4S)-4-amino-N-(propan-2-yl)-1-[2-(pyridin-3-yloxy)acetyl]pyrrolidine-2-carboxamide
7-fluoro-N-(2-hydroxyethyl)-2-methyl-N-[(2-methylphenyl)methyl]quinoline-4-carboxamide
N-(6-phenoxypyridin-3-yl)-1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidine-4-carboxamide
methyl 5-[(butan-2-yl)amino]-3-cyclobutaneamido-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(dimethylamino)-8-(2-phenylpropyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(2-methylphenyl)ethan-1-one
7-(4-chlorophenyl)-2-[(propane-2-sulfonyl)methyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one