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4-methyl-2-{4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl}-6-(trifluoromethyl)pyrimidine
1-[2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidine-3-carboxamide
3-{[4-(2-chlorophenoxy)piperidin-1-yl]methyl}-4-methoxyphenol
5-cyclopropyl-3-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1,2-oxazole
N-[2-(1H-imidazol-1-yl)ethyl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-3-amine
4-({3-methoxy-4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)thiomorpholine
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
(5S,9aS,9bS)-5-[4-(cyclopentyloxy)phenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[1-(dimethylsulfamoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
6-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-N-(propan-2-yl)pyrimidin-4-amine
N-(4-{4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
9-(cyclopropylmethyl)-1-methyl-4-[(3-methylpyridin-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-amino-4-[2-(difluoromethoxy)phenyl]-6-(2-hydroxypropan-2-yl)pyridine-3-carbonitrile
(4aR,7aS)-1-propyl-4-(quinoline-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(2,5-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methylpropanamide
3-({[(5-amino-1,3,4-thiadiazol-2-yl)methyl]carbamoyl}amino)-N-(2-methoxyethyl)-2-methylbenzamide
(3R,4R)-3-methyl-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(oxan-4-yl)piperidin-4-ol
2-(5-acetylthiophen-3-yl)-N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
[(2,6-difluoro-3-methylphenyl)methyl][(3-ethyl-1,2-oxazol-5-yl)methyl]methylamine
3-(2-methoxyphenyl)-3-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)pyrrolidine-2,5-dione
3-acetamido-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}propanamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
1-{2-[1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
(4aS,7aR)-1-(dimethyl-1,3-oxazole-4-carbonyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-chloro-6-methyl-N-[(5-methylpyrazin-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-9-methoxy-7-oxo-N-(thiophen-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-chloro-N-(2-{[3-(2-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}ethyl)benzamide
1-(4-chloro-2-fluorobenzoyl)-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
4-(1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)pyridine
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[4-(trifluoromethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
7-(2-methoxyethyl)-2-(quinoxaline-5-carbonyl)-2,7-diazaspiro[4.5]decane
(3S,9aR)-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-3-propyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(1R,3s,6r,8S)-4-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
(3-benzyl-1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}piperidin-3-yl)methanol
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N2,N2,6-trimethyl-N4-[2-(3-methylpiperidin-1-yl)ethyl]pyrimidine-2,4-diamine
(3S,4R)-4-(3-methoxyphenyl)-1-[3-(methylsulfanyl)propyl]pyrrolidine-3-carboxylic acid
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
5-ethyl-5-{1-[(2-hydroxynaphthalen-1-yl)methyl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
1-({4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)-1H-1,3-benzodiazole
1-({2-[4-(1H-imidazol-1-yl)butoxy]phenyl}methyl)-2-methyl-1,4-diazepan-5-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-[2-(propan-2-yl)pyrimidine-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-(quinoxalin-2-yl)pyrrolidin-3-yl]acetamide
(3S,4R)-4-methyl-1-[2-(morpholin-4-yl)benzoyl]piperidine-3,4-diol