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1-{[2-(carboxymethoxy)-5-chlorophenyl]methyl}-3-ethylpiperidine-3-carboxylic acid
3-ethyl-1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(dimethyl-1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N,2,7,8-tetramethyl-N-[2-(2-oxopiperidin-1-yl)ethyl]quinoline-4-carboxamide
8-(2,6-dimethylhept-5-en-1-yl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-methyl-6-(4-{[4-(4-methylphenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidin-2-amine
N-{2-[1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
3-(3-chloro-1,2-oxazol-5-yl)-N-(thiolan-3-yl)propanamide
3-(4-phenoxybenzoyl)piperidine
1-[(2-fluorophenyl)methyl]-N-[2-(3-methylthiophen-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
N-{1-[7-(furan-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-3-methylbutyl}-3,5-dimethylbenzamide
(3S,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-methylpiperidine-3,4-diol
N-[2-(4-fluorophenyl)ethyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-{1-benzyl-3-[(1,3-thiazol-2-ylmethyl)carbamoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propanoate
4-{pyrazolo[1,5-a]pyrimidin-3-yl}benzamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2-phenoxyethyl)butanamide
3-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
[1-(3-phenylbenzoyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
(1S,5R)-3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-(butylsulfanyl)-6-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrimidin-4-amine
1-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-[(3,3-dioxo-1,3λ6,4-oxathiazinan-4-yl)methyl]-N,N-dimethylfuran-2-carboxamide
4-(propan-2-yl)-6-[3-(propoxymethyl)pyrrolidin-1-yl]pyrimidine
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(3-phenylpropyl)acetamide
2-(4-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
(1S,5R)-3-benzoyl-6-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(4aR,8aS)-1-(2-methoxyethyl)-6-[(4-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-phenoxybutanamide
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
1-[2-(pyridin-2-yl)pyrrolidin-1-yl]-2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethan-1-one
2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-(propan-2-yl)acetamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
2-{2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
{1-[2-(3-phenylpropyl)-1,3-benzoxazole-5-carbonyl]piperidin-2-yl}methanol
1-[2-ethoxy-5-(trifluoromethyl)phenyl]-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
6-cyano-N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methylpyridine-3-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3-methylbenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-methylbenzamide
{1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[1-(2-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]propan-1-one
(2R)-2-amino-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-4,4-dimethylpentanamide
N-methyl-3-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-2-ylmethyl)-5-(2,3,4-trimethoxyphenyl)benzamide
2,5-dimethyl-N-[1-(3-phenylpropyl)piperidin-3-yl]furan-3-carboxamide
2-(3-hydroxypropyl)-9-(naphthalen-1-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[2-(dimethylamino)ethyl]-5-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
N'-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}butanediamide
4-{4-[2-(hydroxymethyl)-4-methylpiperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
(2S)-4-methyl-1-[(1-methyl-1H-pyrazol-5-yl)methyl]-2-phenylpiperazine
2-chloro-6-methoxy-3-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)phenol
1-{3-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one