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5-methoxy-3-(pyridin-3-ylmethyl)-3,4-dihydroquinazolin-4-one
5-(2-chloro-4-methoxyphenoxymethyl)-N-methyl-N-(thiophen-2-ylmethyl)-1H-pyrazole-3-carboxamide
methyl 2-{[2-(pyridin-2-yl)pyrrolidin-1-yl]sulfonyl}benzoate
3-phenyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-pyrazole-4-carboxamide
4-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-3-ethyl-1H-pyrazole
6-methyl-3-[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
3-cyclopropyl-5-{[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole
N-(adamantan-1-yl)-2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
3-[4-(dimethylamino)phenyl]-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
7-[2-(1H-imidazol-1-yl)propanoyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-propylurea
N-[1-(1H-indol-2-yl)ethyl]-N-methyl-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
3-[1-(2-chlorobenzoyl)piperidin-4-yl]-N-[(4-fluorophenyl)methyl]propanamide
1-(2-ethylpyridine-4-carbonyl)-4-(2-methoxyphenyl)-2-methylpiperazine
4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-11-({[3-(trifluoromethyl)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
[(3R,4S)-1-[(2-methyl-1-benzothiophen-3-yl)methyl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-benzyl-1-methyl-N-[(4-methyl-1,3-thiazol-5-yl)methyl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-[4-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)phenyl]imidazolidine-2,4-dione
7a-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}-hexahydro-1H-pyrrolizine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[7-(methylsulfanyl)-2-(morpholin-4-yl)quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
(4aS,7aR)-1-[5-(hydroxymethyl)furan-2-carbonyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-3-[4-(2-methylphenyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)acetamide
N,N-dimethyl-2-(4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)acetamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
N-(cyclopropylmethyl)-1-(prop-2-en-1-yl)-N-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,6-trimethylquinoline-4-carboxamide
5-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
3-(2,3-dimethoxyphenyl)-1-[3-(methylsulfanyl)propyl]pyrrolidine
{3-[5-(2,2-dimethyloxan-4-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-3-(1,2-oxazinan-2-yl)propanamide
3-(4-{5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenyl)propanoic acid
1-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
N-({7-[(3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methylbutanamide
4-[(3-methylphenyl)sulfanyl]-1-(1,2-oxazole-5-carbonyl)piperidine
(3aR,6aR)-N-[(2,6-difluoro-3-methoxyphenyl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-5-methyl-4-(thiophen-2-yl)pyrimidine
N,2-dimethyl-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrido[2,3-d]pyrimidin-4-amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
2-cyclohexyl-5-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)pyrimidine
2-amino-6-(3-methoxyphenyl)-4-(oxolan-3-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-oxo-2H-chromene-3-carboxamide
N-butyl-4-chloro-1,3-dimethyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
7-cyclohexyl-2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
3-cyclobutyl-4-(5-ethylfuran-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N,N-diethyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)[(5-ethylpyridin-2-yl)methyl]amine
4-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-1-phenylpiperazin-2-one
methyl 4-oxo-4-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]butanoate
N-butyl-2-{1-[3-(4-hydroxyphenyl)phenyl]-N-methylformamido}acetamide