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1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
3-[3-(dimethylamino)propyl]-5-{1-[(3,5-dimethylphenyl)methyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]imidazolidine-2,4-dione
(4aR,7aS)-1-ethyl-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)oxane-2-carboxamide
5-[9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
(2R,4S)-4-hydroxy-1-(4-phenylbutanoyl)piperidine-2-carboxylic acid
2-{[(2R)-1-hydroxy-3-methylbutan-2-yl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(3,4-dimethoxyphenyl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(1S,5R)-3-benzoyl-6-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
(1S,9aR)-1-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-octahydro-1H-quinolizine
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-3-(4-methylphenyl)propan-1-one
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
2-[({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]-1-(morpholin-4-yl)ethan-1-one
3-[(4-fluorophenyl)methyl]-N-[1-(4-methoxyphenyl)ethyl]-N-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(2-aminoethyl)-N,5,6-trimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
3-[2-(1-{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]phenol
2-(2,5-difluorophenyl)-5-(1H-imidazol-1-ylmethyl)pyridine
3-{imidazo[1,2-a]pyridin-2-yl}-1-[3-(phenylamino)piperidin-1-yl]propan-1-one
1-[1-(cyclohex-1-en-1-yl)ethyl]-3-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
(2S)-2-(hydroxymethyl)-N-[2-(4-methoxyphenyl)phenyl]pyrrolidine-1-carboxamide
2-methyl-6-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2,3-dihydropyridazin-3-one
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine
1-ethyl-5-{[4-(3-phenyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1H-1,2,4-triazole
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
3-{1-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-imidazol-2-yl}pyridine
1-methyl-5-phenyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-pyrazole-3-carboxamide
N-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-carboxamide
3-[5-(2,6-dimethyl-1H-indol-3-yl)-4-phenyl-1H-imidazol-1-yl]propane-1,2-diol
(1R,2S,6R,7S)-4-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-4-azatricyclo[5.2.2.02,6]undecane
2-(2-methoxyethoxy)-1-[3-(3-methylphenyl)piperidin-1-yl]ethan-1-one
N2-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-N4-methylpyrimidine-2,4-diamine
2-amino-3-ethyl-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[3-(2-chlorophenyl)phenoxy]propanamide
6-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
4-(dimethyl-1,3-thiazole-5-carbonyl)-1-(1H-indazol-5-yl)piperazin-2-one
1-[4-(4-fluorophenoxy)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
3-{1-[(4-ethoxyphenyl)methyl]piperidin-3-yl}-N-(4-fluoro-2-methylphenyl)propanamide
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(thiophen-2-yl)propan-1-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-propylpyridine-4-carboxamide
N-[(2-ethoxyphenyl)methyl]-2-oxo-N-(prop-2-en-1-yl)-1-oxaspiro[4.4]nonane-4-carboxamide
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[3-(methylsulfanyl)phenyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-benzyl-8-[(2,6-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[4-(3,4,5-trimethoxyphenyl)phenyl]-1H-pyrazole
3-(7-chloroquinoxalin-2-yl)-3,9-diazaspiro[5.6]dodecan-10-one
1-[2-amino-4-(3-hydroxypyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-2-(2-phenylethyl)morpholine
6-(morpholin-4-yl)-N4-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrimidine-2,4-diamine
N-methyl-2-{4-[({[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}carbamoyl)amino]phenyl}acetamide
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-5,6,7,8-tetrahydroquinoline