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9-methyl-3-(3,3,3-trifluoropropanesulfonyl)-3,9-diazaspiro[5.6]dodecane
(2R,3R,6R)-3-phenyl-5-[3-(pyridin-3-yl)propyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}-2,6-dimethylphenol
5-[butyl(methyl)amino]-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-(cyclohexylmethyl)-4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
5-methyl-N-({3-methyl-7-[2-(phenylsulfanyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)pyrazine-2-carboxamide
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3-(thiophene-2-carbonyl)piperidine
N-[5-(furan-2-yl)-1,3,4-thiadiazol-2-yl]-4-(pyridin-2-yl)piperazine-1-carboxamide
(3S,7S,8aS)-7-{[(4-chlorophenyl)methyl]amino}-3-(1H-indol-3-ylmethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
5-ethyl-1'-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-4-(pyrrolidine-1-carbonyl)piperidine
2-{[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]amino}-N-[(2-fluorophenyl)methyl]acetamide
1-[(4-fluoro-2-methylphenyl)methyl]-4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-methoxy-6-[(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)methyl]phenol
(4aS,8aR)-6-(2,5-dimethylfuran-3-carbonyl)-1-(4-hydroxybutyl)-decahydro-1,6-naphthyridin-2-one
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
3-(2H-1,3-benzodioxol-5-yl)-1-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methylurea
(2S)-N-[(3-ethoxy-4-methoxyphenyl)methyl]piperidine-2-carboxamide
3-(2-methoxyethyl)-1-(pyridin-3-ylmethyl)piperidine-3-carboxylic acid
ethyl 4-(2-methoxyethyl)-1-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-ylmethyl}piperidine-4-carboxylate
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(pyridin-3-yloxy)propyl]-1H-pyrazole-4-carboxamide
2-[(4-methoxyphenyl)methyl]-4-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[2-(dimethylamino)ethyl]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
8-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-ethyl-2,8-diazaspiro[4.5]decan-3-one
2-(4-acetylphenoxy)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylacetamide
2-methyl-N-{1-[7-(naphthalen-1-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
3-hydroxy-N-{1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl}propanamide
(3S)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-N,N-dimethylazepan-3-amine
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-2-carboxamide
6-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-(3-hydroxyphenyl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-3-methoxypropanamide
2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-{[(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
{2-[(1H-1,3-benzodiazol-2-ylmethyl)(thiophen-3-ylmethyl)amino]ethyl}dimethylamine
(4aR,8aS)-1-[2-(4-methoxyphenyl)ethyl]-6-[(1-methyl-1H-pyrrol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
3-(2-methyl-1H-imidazol-1-yl)-1-[3-(3-methylphenoxymethyl)piperidin-1-yl]propan-1-one
3-{[(4aS,7aR)-6,6-dioxo-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-methoxybenzamide
methyl (1R,3S,3aR,6aS)-1-methyl-3-(3-methylthiophen-2-yl)-4,6-dioxo-5-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
3-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-(2-methylpropyl)-1,2,4-oxadiazole
1-[(2-fluorophenyl)methyl]-N-[1-(6-methoxynaphthalen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(5-fluoro-2-methoxybenzoyl)-1-(3-phenylprop-2-yn-1-yl)piperidine
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
5-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-4-(trifluoromethyl)pyrimidin-2-amine
1-{4-[2-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)quinazolin-4-yl]piperazin-1-yl}ethan-1-one
4-[4-(2-methoxyphenyl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
2-(dimethylamino)-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(3aS,6aR)-5-benzyl-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one