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5-(2,6-dimethoxyphenyl)-3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1,2,4-triazine
5-ethyl-2-(4-{[4-(1-hydroxypropyl)piperidin-1-yl]methyl}phenyl)-6-methyl-3,4-dihydropyrimidin-4-one
(3S,4S)-4-methyl-1-{[2-(propylamino)pyrimidin-5-yl]methyl}piperidine-3,4-diol
N-cyclopentyl-2-[(2-phenoxyethyl)amino]propanamide
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
5-methyl-5-{1-[2-(2-methyl-1H-indol-3-yl)acetyl]piperidin-4-yl}-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-3-(2-methyl-1H-indol-1-yl)propanamide
1-{[4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine
2-oxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-6-(pyrrolidin-1-ylmethyl)-1,2-dihydropyridine-3-carboxamide
6-[3-(1H-indazol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(2,5-dimethylphenyl)-2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}acetic acid
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}oxan-4-amine
N-[2-(dimethylamino)ethyl]-2-methoxy-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
(2S)-2-{[(cyclooctylcarbamoyl)methyl]amino}-3-phenylpropanamide
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(2-fluorophenyl)propan-1-one
methyl 4-[2-amino-3-cyano-6-(propan-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl]thiophene-2-carboxylate
1-[2-(dimethylamino)-6-(oxolan-3-ylmethyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-4-yl]piperidin-4-ol
4-[(2-chloro-4-fluorophenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
2-methyl-8-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
{[1-(1-cycloheptylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}(ethyl)(propan-2-yl)amine
N2-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-N1-(pyridin-3-yl)ethane-1,2-diamine
1-[4-(2-methoxyphenyl)piperazin-1-yl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
2,3-dimethyl-7-[3-(1H-pyrazol-4-yl)benzoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
5-methyl-1-(4-methylphenyl)-4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
4-chloro-3-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1H-pyrazol-5-amine
(3S,4S)-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-[(1-hydroxycyclohexyl)methyl]-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
N-[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-(2-oxopyrrolidin-1-yl)benzamide
(4aR,8aR)-7-(4-cyanopyridin-2-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
3-(2-amino-1,3-thiazol-4-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
1-(4-methylphenyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(2S)-2-(methoxymethyl)-N-[4-(thiophen-2-ylmethoxy)phenyl]pyrrolidine-1-carboxamide
1-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-4-yl)piperidin-3-ol
N,N-dimethyl-2-[(1S,5R)-7-oxo-3-[6-(propan-2-yl)pyrimidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
1-[4-({4-[(2,6-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
2-(2-hydroxyethyl)-N-[2-methyl-4-(propylcarbamoyl)phenyl]-3-oxopiperazine-1-carboxamide
2-(1-methyl-4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]propanamide
3-[2-(2-ethylpiperidin-1-yl)-2-oxoethyl]-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3-(dimethyl-1,2-oxazol-4-yl)propanamide
3,5-dimethyl-2-[({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]pyridin-4-ol
N-[(2-chlorophenyl)methyl]-6-{[(2-hydroxy-2-phenylethyl)(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
3-{5-[2-(2-methoxyphenyl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
4-(2-amino-6-methylpyrimidin-4-yl)-7-(5-chloropyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-chloro-5-({3-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine
N-methyl-5-(phenoxymethyl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrazole-3-carboxamide
3-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1-(2-hydroxypyridin-3-yl)urea
1-[(2-chloro-6-fluorophenyl)methyl]-3-[2-(methylsulfanyl)ethyl]-5-(oxolan-3-yl)-1H-1,2,4-triazole
5-(morpholin-4-ylmethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]furan-3-carboxamide