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6-({[(5-chloro-1-benzothiophen-3-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)pyrazin-2-amine
N-(2-methyl-1,3-benzothiazol-5-yl)-4-(3-methylpyridin-2-yl)piperazine-1-carboxamide
5-[(3-phenoxyphenyl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
(2S,4S)-4-amino-1-[4-(diethylamino)benzoyl]-N-methylpyrrolidine-2-carboxamide
3-[1-(5-chloro-3-phenyl-1H-indol-2-yl)-N-methylformamido]-N-methylpropanamide
(3R,5R)-N-butyl-1-[(4-hydroxyphenyl)methyl]-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
1-methyl-4-[4-(trifluoromethyl)pyrimidin-2-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[3-(2-chlorophenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-indazol-3-yl)acetamide
6-methyl-3-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane-8-carbonyl}-1,2-dihydropyridin-2-one
3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1-methyl-1-[3-(1-methyl-1H-imidazol-2-yl)propyl]urea
4,4,4-trifluoro-1-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidin-1-yl]butan-1-one
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-ethoxy-5-[2-(furan-2-yl)pyrimidin-4-yl]benzoic acid
5-(phenoxymethyl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-methyl-2-(1-{[5-methyl-2-(naphthalen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl][2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]methylamine
{[2-(difluoromethoxy)phenyl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
6-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
1-{1-[(2,4-dimethoxy-3-methylphenyl)methyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
2-{1-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-1H-1,2,3-triazol-4-yl}benzoic acid
N-{1-azabicyclo[2.2.2]octan-3-yl}-1-benzofuran-3-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
3-(4-chloro-2-methylbenzoyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidine
1-{2-[4-(hydroxymethyl)piperidin-1-yl]ethyl}-3-[2-(3-methylphenoxy)phenyl]urea
4-(3-methoxypyrazin-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(2-phenylethyl)-1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine
7-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-[2-(pyridin-3-yloxy)propyl]-1,4-dithiepan-6-amine
(1R,3S)-7-(6-methylpyridine-2-carbonyl)-7-azaspiro[3.5]nonane-1,3-diol
2-(3-methoxybenzenesulfonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]acetamide
N-cyclohexyl-1-cyclopropyl-5-[4-(4-methylphenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2-methoxy-4-[(1E)-pent-1-en-1-yl]pyridine-3-carbonitrile
N,N-dimethyl-2-[({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]acetamide
5-(2H-1,3-benzodioxol-5-yl)-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1,2,4-triazin-3-amine
N-methyl-N-[2-(methylsulfanyl)ethyl]-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
1-{[3-(cyclopentyloxy)phenyl]methyl}piperidine-4-carbonitrile
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-methylpyridine
N-(2-{4-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]morpholin-2-yl}ethyl)acetamide
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}(2,3-dihydro-1-benzofuran-2-ylmethyl)methylamine
N-{1-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylthiophene-3-carboxamide
(3S)-4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,3-dimethylpiperazin-2-one
5-(4-hydroxypiperidin-1-yl)-N-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{2-[1-(3-hydroxy-2-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
6-[3-(hydroxymethyl)piperidin-1-yl]-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
8-(6-aminopyrimidin-4-yl)-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(3S,4R)-1-(5-cyanopyridin-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide