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4-{2-methyl-6-[1-(pyridine-4-carbonyl)piperidin-3-yl]pyrimidin-4-yl}morpholine
2-[2-(methylsulfanyl)phenyl]-2-[4-(pyridin-3-ylmethyl)piperazin-1-yl]acetic acid
3-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
(3aR,7aS)-N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
1-[3-(5-methylfuran-2-yl)butyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
8-(6-hydroxy-1,4-diazepan-1-yl)-3,7-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dione
6-methyl-1-{3-oxo-3-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]propyl}-1,2-dihydropyridin-2-one
1-(3-{6-[(2-hydroxyethyl)amino]pyridazin-3-yl}phenyl)ethan-1-one
dimethyl({4-[3-methyl-1-(propan-2-yl)-1H-pyrazol-4-yl]phenyl}methyl)amine
[3-(2-phenoxyethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl]methanol
1-{1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]piperidin-4-yl}-3-methylbutan-1-ol
2-(2,2,2-trifluoroethanesulfonyl)-2,8-diazaspiro[4.5]decane
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]piperidine-3-carboxamide
N-[(3-fluoro-4-methoxyphenyl)methyl]-N-(3-methoxypropyl)-1-methylpiperidin-4-amine
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[(4-methyl-1,3-thiazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-fluoroethyl)-3-({1-oxaspiro[4.4]nonan-3-yl}sulfamoyl)benzamide
2-[1-(cyclohexylmethyl)-4-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-[(3-methylpyridin-4-yl)methyl]pyridin-2-amine
(3S)-3-benzyl-4-[(5-fluoro-2-methoxyphenyl)methyl]piperazin-2-one
2-(adamantan-1-yl)-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]acetamide
N-[(3S,4R)-1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
methyl 3-[1-(4-chlorophenyl)cyclopropaneamido]-5-{[(4-methyl-1,2,5-oxadiazol-3-yl)formamido]methyl}benzoate
methyl 2-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}benzoate
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-4-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
3-[4-methyl-2-(2,3,4-trimethoxyphenyl)phenyl]-1,3-oxazolidin-2-one
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(pyridin-4-ylsulfanyl)acetamide
(3S,4R)-3-benzyl-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-methylpiperidin-4-ol
N,4-dimethyl-2-(methylamino)-N-[(3-methylpyridin-4-yl)methyl]-1,3-thiazole-5-carboxamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-propylbenzamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-2-(2-methoxyethyl)morpholine
5-{1-[2-(quinazolin-4-yloxy)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
3-benzyl-8-[(3-hydroxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(4-fluoro-2-methylphenyl)-2-{[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]amino}acetamide
5-[1-(4-chloro-1H-pyrazol-1-yl)ethyl]-1-[(3-methoxyphenyl)methyl]-1H-1,2,4-triazole
3-(2-methoxyphenyl)-N-[1-({[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
4-({2-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
(3S,9aR)-3-[(2S)-butan-2-yl]-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-(1-methyl-1H-imidazole-5-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(4-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}phenyl)piperidine
(4aR,7aS)-1-methyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 3-{[(2,2-dimethyloxan-4-yl)formamido]methyl}-5-(2-methoxybenzamido)benzoate
1-{[5-(methoxymethyl)furan-2-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(4-fluorophenoxymethyl)piperidine
1-(furan-2-ylmethyl)-2-(pentan-2-yl)-1H-imidazole
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-7-oxo-3-(2,2,3,3-tetramethylcyclopropanecarbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2,3-difluoro-N-(2-hydroxyethyl)-4-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
N-(1,3-benzothiazol-2-ylmethyl)-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-benzyl-8-(1-ethyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)propyl]-3-(3-methylphenyl)piperidine