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4-ethyl-3-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
(2E)-N-[(3-methyl-7-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-phenylprop-2-enamide
1-methyl-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(azepan-1-yl)-1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}ethan-1-one
(2R,4S)-1-[(3E)-hex-3-enoyl]-4-hydroxypiperidine-2-carboxylic acid
N3-[(6-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N5-(cyclohexylmethyl)-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]-N-(pyridin-3-yl)propanamide
2-(2-{4-[1-(2,3-dihydro-1H-inden-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)pyridine
2-[2-(1H-imidazol-4-yl)ethyl]-8-[3-(1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
3-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-(pyrrolidin-1-yl)propan-1-one
1-(4-chlorophenyl)-N-{[1-(pyridin-2-ylmethyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
1-cyclohexyl-4-{6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carbonyl}piperazin-2-one
5-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N,3,5-trimethyl-N-(2-phenylethyl)-1-benzofuran-2-carboxamide
6-methyl-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-phenylpropyl)piperidine-4-carboxamide
(1S,5R)-6-[(2,6-difluoro-3-methylphenyl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-[(3-methyloxetan-3-yl)methyl]-1-(2-propylphenyl)urea
(4aS,7aR)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-cyclobutanecarbonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-phenylpropyl)-4-[(pyridin-2-ylmethyl)amino]pyrrolidin-2-one
methyl 5-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-5-oxopentanoate
(2R,3R)-3-[4-(4-chlorophenyl)-1H-1,2,3-triazol-1-yl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-butoxy-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyridin-2-amine
(2S,4S)-4-amino-N-ethyl-1-{pyrazolo[1,5-a]pyridine-2-carbonyl}pyrrolidine-2-carboxamide
N-[2-(1H-indol-1-yl)ethyl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-(4-ethylpiperazin-1-yl)-N-[1-(pyridin-2-yl)propan-2-yl]-2,3-dihydro-1H-indene-2-carboxamide
methyl 4-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperazine-1-carboxylate
N-[(3-methoxyphenyl)methyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
(3S,4R)-1-(3-fluoropyridin-2-yl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
4-(1-ethylpiperidine-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
7-[(2,3-difluorophenyl)methyl]-2-(furan-3-carbonyl)-2,7-diazaspiro[4.5]decane
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-(4-benzylpiperidin-1-yl)propan-1-one
2-benzyl-9-[(2S)-2,3-dihydroxypropyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 3-[(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazol-4-yl)formamido]propanoate
4-[1-(3-phenylpropyl)-5-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[(3S,4S)-3-hydroxy-4-(pyrrolidin-1-yl)pyrrolidin-1-yl]ethan-1-one
5-(propan-2-yl)-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
N-ethyl-N-(pyridin-4-ylmethyl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-amine
(4aR,7aS)-N-[4-(1H-imidazol-1-yl)phenyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
3-{[(3R,5S)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}-1-methyl-1,2-dihydroquinolin-2-one
(1R,3S)-7-[2-hydroxy-3,5-bis(propan-2-yl)benzoyl]-3-methoxy-7-azaspiro[3.5]nonan-1-ol
(4aS,8aR)-6-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
2-[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]-1,3-thiazole-4-carboxamide
(3S,4S)-4-cyclopropyl-1-[3-(4-methylphenyl)propanoyl]pyrrolidine-3-carboxylic acid
(4aS,8aR)-2-{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}-decahydroisoquinoline
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(furan-2-yl)ethyl]piperidin-4-amine
N-methyl-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
7-[(4-fluorophenyl)methyl]-2-(2-methylpropyl)-2,7-diazaspiro[4.5]decan-6-one