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N,6-dimethyl-2-[(2-methylphenyl)methyl]-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(4aS,8aR)-6-(2-methylpyrimidin-4-yl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
2-(1H-1,3-benzodiazol-1-yl)-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}acetamide
6,8-dimethyl-3-({8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1,2-dihydroquinolin-2-one
4-[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-(pyridin-3-ylmethyl)pyrimidin-2-amine
3-{2-[2-(furan-2-yl)azepan-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
5-cyclopropyl-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-1,3-oxazole-4-carboxamide
1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
4-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-[2-(methylsulfamoyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(2S)-2,6-diamino-1-[4-(4-methylphenoxy)piperidin-1-yl]hexan-1-one
1-{[2-(3-fluorophenoxymethyl)-6-oxo-1,6-dihydropyrimidin-4-yl]methyl}-3,3-dimethylurea
4,4-difluoro-1-({2-[2-(3-methylpiperidin-1-yl)ethoxy]phenyl}methyl)piperidine
N3-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N5-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-(3-methoxypropyl)-2-(2-methyl-5-oxopyrrolidin-1-yl)-N-[(4-methylphenyl)methyl]acetamide
2-{3-[1-(3-methoxypropyl)-1H-pyrazol-3-yl]phenyl}pyrazine
2-(3-methylbutyl)-8-(4-propyl-1,2,3-thiadiazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
2-(cyclohexylmethyl)-4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)morpholine
2-(4-{2-[(3-fluoro-4-methylphenyl)methyl]benzoyl}morpholin-3-yl)acetamide
5-(methoxymethyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
ethyl 5-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
5-(2,4-difluorophenoxymethyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
3-(4-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazin-1-yl)propan-1-ol
3-[5-(propylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N,2-dimethyl-N-[2-(morpholin-4-yl)propyl]-6-(propan-2-yl)pyrimidin-4-amine
7-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[2-(ethylsulfanyl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-(2-methylpropyl)-5-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
2-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-ethyl-5-[1-(furan-3-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-1H-1,2,4-triazole
4-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}-5-methyl-1-(2-methylphenyl)piperazin-2-one
N-{[4-benzyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
butyl 3-{[(2-chlorophenyl)formamido]methyl}piperidine-1-carboxylate
4-{5-[1-(5-methyl-1,3-oxazole-4-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}thiomorpholine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-methanesulfonyl-2-methylpyrimidin-4-amine
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
4-{[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]methyl}benzamide
2-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]amino}pyridine-4-carboxamide
N-(4-fluorophenyl)-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-amine
2-methyl-4-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-1,3-thiazole
2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
2-methyl-5-({3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[(5-methylpyrazin-2-yl)methyl]acetamide
2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetic acid
3-{1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide
5-(2,6-dimethoxyphenyl)-N-[3-(1H-indazol-1-yl)propyl]-1,2,4-triazin-3-amine