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4-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}piperazine-1-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(ethanesulfonyl)-2,7-diazaspiro[4.5]decane
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[4-(trifluoromethyl)phenyl]methyl}amine
N-(2,2-dimethyloxan-4-yl)-2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]acetamide
1-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
N-[1-(propan-2-yl)cyclopropyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-tert-butyl-4-(4-{[4-(propan-2-yl)piperidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
(1-{2-[(5-methylpyrimidin-2-yl)amino]ethyl}piperidin-4-yl)methanol
N-(1-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
2-methoxy-N-[1-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-1-[4-(2-ethoxyphenyl)piperazin-1-yl]propan-1-one
4-{3-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
3-(2H-1,3-benzodioxol-5-ylmethyl)-3H,4H-pyrido[2,3-d]pyrimidin-4-one
2-(4-chlorophenyl)-4-(1H-pyrrole-2-carbonyl)morpholine
4-(3-methyl-1H-pyrazole-4-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
1-{5-[(5,6-dimethylpyrimidin-4-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
4-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-5-ethylpyrimidin-2-amine
1-[1-(3-{thieno[2,3-d]pyrimidin-4-yl}phenyl)ethyl]pyrrolidine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-methyl-1H-indol-1-yl)propanamide
N-(2-hydroxypropyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
methyl({[5-(6-methylpyridazin-3-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-(propan-2-yl)pyrimidin-4-amine
N-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2,5-dihydro-1H-pyrrole-2-carboxamide
1-[2-(dimethylamino)ethyl]-N,3-dimethyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
2-amino-6-cyclopropanecarbonyl-4-[4-(methylsulfanyl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-4-oxobutanamide
3-[4-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperazin-1-yl]-2,5-dimethylpyrazine
(2E)-N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
7-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decane
7-(1,3-benzothiazol-2-yl)-4-[(4-fluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2S,4R)-4-amino-N-ethyl-1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)pyrrolidine-2-carboxamide
N-[4-(4-{[3-(2-methoxyphenyl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]furan-3-carboxamide
7-acetamido-1-ethyl-2-(2-fluorophenyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-{1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-4-methyl-1H-1,3-benzodiazole
N-[4-(pyridin-2-yl)butyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-(3-fluoro-4-methoxybenzoyl)-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]propan-1-one
8-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
3-{2-[({4-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)amino]ethyl}-1,3-oxazolidin-2-one
4-{3-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]butyl}morpholine
N-[(3,4-dimethoxyphenyl)methyl]-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]isoquinoline
N-(2,3-dihydro-1H-inden-2-yl)-4-[(4-methoxy-3-methylphenyl)methyl]morpholine-2-carboxamide
4-{2-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1-(propan-2-yl)-1H-pyrazole
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
1-cyclohexyl-1-(pyridin-3-ylmethyl)-3-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
[(1,3-dimethyl-1H-pyrazol-5-yl)methyl][(5-methylthiophen-2-yl)methyl](prop-2-en-1-yl)amine
(4aR,7aS)-1-cyclopropanecarbonyl-4-[(3,4-dimethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(1R,5R)-6-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide