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(1S,5R)-3-[(4-methoxy-3-methylphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N,2-dimethyl-N-[2-(piperidin-1-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[(3,5-dimethylphenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-one
4-{[(6-methoxypyrimidin-4-yl)amino]methyl}benzene-1-sulfonamide
1-(3-methylbutyl)-N3-(2-methylpropyl)-N5-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(2R,3R,6R)-5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(2-fluorophenyl)methyl]-N-{spiro[2.5]octan-1-ylmethyl}-1H-1,2,3-triazole-4-carboxamide
2-amino-N-[1-(3-fluoro-4-methoxyphenyl)ethyl]-4-phenylpyrimidine-5-carboxamide
5-(1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(3-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-ethyl-6-{4-[4-(4-methoxybutyl)piperazin-1-yl]piperidin-1-yl}-2-methylpyrimidine
8-[2-(3-hydroxyphenyl)acetyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(2-fluorophenoxy)-N-(2,4,6-trimethylpyridin-3-yl)azetidine-1-carboxamide
N-[(3R,4S)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
3-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
3-[3-(2-methyl-1,3-thiazol-4-yl)-5-[(methylamino)methyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
3-[4-(3-methyl-5-propyl-1-benzofuran-2-carbonyl)piperazin-1-yl]-1λ6-thiolane-1,1-dione
3-(4-methyl-1,3-thiazol-5-yl)-1-[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
(2-methoxyethyl)({[2-(propan-2-yl)pyrimidin-4-yl]methyl})(thiophen-2-ylmethyl)amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}cyclobutan-1-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(5-fluoro-2-methylphenyl)acetamide
N-cyclopropyl-1-(2-ethoxyethyl)-N-(2-methylpropyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3aR,6aR)-2-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-methyl-2-phenyl-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}propanamide
methyl 8-(1-benzyl-1H-pyrazole-4-carbonyl)-1-methoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
(3S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
5-propyl-4-(pyridin-4-yl)thiophene-2-carboxylic acid
4-acetyl-N-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-1,4-diazepane-1-carboxamide
2-amino-4-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-6-(1H-pyrrol-3-yl)pyridine-3-carbonitrile
N-({5-[(2-fluoro-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
2-(3-{[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]methyl}phenoxy)ethan-1-ol
2-(methoxymethyl)-5-[1-(5,6,7,8-tetrahydronaphthalen-1-yl)-1H-imidazol-2-yl]pyrimidine
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(5S,9aS,9bS)-2-phenyl-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(3-methylthiophen-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-methyl-N-{2-[4-({methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)phenoxy]ethyl}-4-(trifluoromethyl)benzamide
2-(1H-pyrazol-1-yl)-1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]butan-1-one
1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-4-(pyridine-4-carbonyl)-1,4-diazepan-2-one
4-{3-[(2-methoxyphenyl)methyl]-5-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}-1-methylpiperidine
8-{4-[4-(2-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2,6-dimethyloctan-2-ol
3-(2-fluorophenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
(1s,4s)-4-{4-[(3Z)-hex-3-en-1-yl]-1H-1,2,3-triazol-1-yl}cyclohexane-1-carboxylic acid
3-methoxy-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-4-(thiophen-2-yl)butan-1-one
3-[1-(methoxymethyl)cyclopentyl]-1-[3-(methylsulfanyl)phenyl]urea
[(2-cyclohexylpyrimidin-5-yl)methyl]({[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})methylamine
N,N-diethyl-1-(2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperidine-4-carboxamide
N-(2-{7-[(3-ethoxy-4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
5-(5-{[(2-ethyl-6-methylpyridin-3-yl)oxy]methyl}-1,2,4-oxadiazol-3-yl)-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-[5-(1-hydroxy-3-methylbutyl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-3-yl]acetamide