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3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N,8-dimethyl-N-(1,2-oxazol-3-ylmethyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-(7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
N'-butyl-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-N'-[(5-methylthiophen-2-yl)methyl]ethanediamide
1-(4-chlorophenyl)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}cyclobutane-1-carboxamide
(7R,8aS)-7-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-3,4-dimethoxybenzamide
2-[1-(2-methanesulfonylethyl)-1H-imidazol-2-yl]-1-(4-methoxyphenyl)-1H-imidazole
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N,3,6-trimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-benzofuran-2-carboxamide
4-[3-(methanesulfonylmethyl)piperidin-1-yl]-2,5,6-trimethylpyrimidine
N-[(1-ethylpyrrolidin-3-yl)methyl]-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
7-(2-hydroxyethyl)-2-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-N-[(8-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]propanamide
N-cyclopropyl-3,6,7-trimethyl-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
5-methyl-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-1H-indazole-3-carboxamide
3,3-dimethyl-1-{2-oxo-2-[(1S,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}urea
1-(azetidin-1-yl)-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)ethan-1-one
3-{4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}propan-1-ol
4-[(2,3-difluoro-4-methylphenyl)methyl]-5-methyl-1-(2-methylphenyl)piperazin-2-one
1-(6-fluoro-4-methylquinazolin-2-yl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}piperidine-4-carboxamide
(2E)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-3-(pyridin-2-yl)prop-2-enamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]urea
methyl 5-(3-acetamidothiophene-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
8-(8-chloro-2-methylquinoline-4-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-[1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)azetidin-3-yl]pyridine
4-[3-(2-oxopyrrolidin-1-yl)benzoyl]-1-phenylpiperazin-2-one
3-({1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-4-yl}oxy)pyridine
5-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridin-2-ol
7-chloro-4-(1-methyl-1H-indole-6-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2R)-4-methyl-2-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamido]pentanamide
3-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)propanamide
3-(2-phenoxyethyl)-8-[1-(1H-pyrazol-1-yl)propan-2-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(2,4-dimethoxybenzoyl)-1-(oxan-4-yl)piperidine
1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-3-[4-(2-methylphenyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
N-(1-acetylpiperidin-4-yl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
6-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
benzyl({[1-(morpholin-4-yl)cycloheptyl]methyl}sulfamoyl)amine
N-[3-(dimethylamino)-1-phenylpropyl]-6-methoxy-3-methyl-1-benzofuran-2-carboxamide
2,3,4-trimethoxy-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzamide
1-[5-(methoxymethyl)thiophene-2-carbonyl]-4-(pyridin-3-ylmethyl)piperazine
8-(2-methoxyacetyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-(2-methylpropanoyl)-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-(naphthalen-2-yl)-1-phenyl-1H-1,2,3,4-tetrazole
N-{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
1-ethyl-4-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
1-(6-chloro-2-methylquinoline-4-carbonyl)-4-(hydroxymethyl)azepan-4-ol
8-[(3-hydroxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione