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2-methoxy-3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyridine
4-(2-methoxyphenoxy)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylic acid
6-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyridine-2-carboxylic acid
1-ethyl-3-(4-methylpiperazine-1-carbonyl)-N-[(1-phenylcyclopentyl)methyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(3-fluorophenyl)-N-{[1-(propan-2-yl)pyrrolidin-2-yl]methyl}benzamide
3-(2-methylphenyl)-N-[(5-methylpyrazin-2-yl)methyl]-3-phenylpropanamide
7-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
2-(4-methyl-1H-1,3-benzodiazol-2-yl)-N-(2-methyl-2H-1,2,3-benzotriazol-4-yl)pyrrolidine-1-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-3-phenylbutanamide
N,N-dimethyl-7-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-ethyl-N-[3-(1H-imidazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
3-(2-chlorobenzoyl)-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)azepan-4-amine
4-({5-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl](methyl)[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
1-[(2-chloro-4-fluorophenyl)methyl]-N-(1H-indol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{1-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-phenylethan-1-one
1-[(3aS,6aS)-5-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-octahydropyrrolo[2,3-c]pyrrol-1-yl]-2-methoxyethan-1-one
2-(cyclopent-2-en-1-yl)-1-[2-ethyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
1-(1-methyl-1H-pyrazole-5-carbonyl)-3-[4-(trifluoromethyl)benzoyl]piperidine
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-[(propan-2-yl)amino]pyrrolidine-2-carboxamide
N-[(3S,4R)-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-4-propylpyrrolidin-3-yl]acetamide
6-[4-(2-fluorophenyl)benzoyl]-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
N-{2-[ethyl(methyl)amino]butyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(1H-imidazol-4-yl)ethyl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
2-ethoxy-6-{[methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amino]methyl}phenol
5-methoxy-2-{[3-(3-methoxybenzoyl)piperidin-1-yl]methyl}phenol
1-(diethylamino)-3-[2-methoxy-5-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
1-(5-chloro-2-methoxyphenyl)-5-cyclopentyl-3-(oxan-4-yl)-1H-1,2,4-triazole
N-[2-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)ethyl]-N-methylmethanesulfonamide
3-{1-[(5-chloro-2-hydroxyphenyl)methyl]piperidin-3-yl}-N-(3,5-dimethoxyphenyl)propanamide
1-cyclohexanecarbonyl-4-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperazine
5-[2-(benzyloxy)phenyl]-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
(1S,6R)-N-[2-(4-fluorophenyl)ethyl]-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
7-cyclopropanecarbonyl-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-[3-(furan-2-yl)propyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-2-(pyridin-3-yl)morpholine
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-acetamido-N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]benzamide
1-(3,5-dichlorophenyl)-3-methyl-3-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]urea
N-[(4,6-dimethylpyridin-2-yl)methyl]-5-ethyl-N-methyl-1,3,4-oxadiazol-2-amine
1-benzyl-5-acetamido-N,2-dimethyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-[2-(1,3-thiazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-1-[(1-phenylpyrrolidin-3-yl)methyl]urea
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-propoxyethan-1-one
3-acetamido-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1-(1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)piperidin-3-ol