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1-(3-fluorophenyl)-3-{1-[1-(1H-indole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
N-(2-fluoroethyl)-3-{6-oxa-9-azaspiro[4.5]decane-9-sulfonyl}benzamide
1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-5-(1,2,5-thiadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-{[7-fluoro-2-(2-methylphenyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-(naphthalen-2-ylmethyl)piperidin-4-ol
(2R,3R,6R)-5-(2-methoxyethyl)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-propyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
7-methyl-3-[(3-phenoxyphenyl)methyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
(2R)-2-hydroxy-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}propan-1-one
3-{[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
methyl[(3-methylquinoxalin-2-yl)methyl][(1-phenyl-1H-pyrazol-4-yl)methyl]amine
(1S,5R)-N,N-dimethyl-6-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
2-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
[3-methyl-9-(1-methylcyclopropanecarbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
(1R,5R)-6-(2-phenylethyl)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[1-(4-methylphenyl)propan-2-yl]-4-(pyridin-4-ylmethyl)-1,4-diazepan-5-one
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(4-methylphenoxymethyl)piperidine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}benzamide
4-{3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}-1-phenylpiperazin-2-one
3-{2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
methyl 3-{[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetamido]methyl}-5-(3-methoxybenzamido)benzoate
4-{3-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenyl}phenol
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
4-[(2S)-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-2-carbonyl]morpholine
[(2S,4R)-1-methyl-4-{2-[5-(2-methylpropyl)thiophen-2-yl]-1H-imidazol-1-yl}pyrrolidin-2-yl]methanol
1-[2-(2-methoxyphenyl)acetyl]-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-(1-tert-butyl-1H-pyrazol-4-yl)-8-methyl-4-(2-methylpyrrolidine-1-carbonyl)quinoline
ethyl 4-[(3-methoxyphenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxylate
1-(2-methoxyphenyl)-4-[1-(3-methylbenzoyl)piperidin-3-yl]piperazine
1-(1-{[5-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}piperidin-4-yl)piperidine-4-carboxylic acid
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]propan-1-one
9-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]-5-(propan-2-yl)-1,2,4-oxadiazole
2-[1-cyclopentyl-4-(1H-pyrazol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
1-{[5-(oxan-2-yl)furan-2-yl]methyl}-4-phenylpiperidine-4-carbonitrile
4-{5-[(2S)-1-(1H-1,2,3-triazole-5-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)acetamide
2-[2-(butan-2-yl)phenoxy]-N-[2-(4-hydroxypiperidin-1-yl)ethyl]acetamide
(1S,5R)-3-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
9-[(3-fluoro-2-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)propanamide
3-(cyclobutylmethoxy)-5-{[(1r,4r)-4-hydroxycyclohexyl]carbamoyl}benzoic acid
1-(5-{[(1,3-benzoxazol-2-ylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(diethylamino)propan-2-ol
1-cyclobutanecarbonyl-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carboxamide
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyridin-3-ylmethyl})amine
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
9-(5-chlorofuran-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]thiomorpholine