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3-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]pyridine
(3S,9aR)-8-[(3-chlorophenyl)methyl]-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(cyclohexylmethyl)-4-(1,3-thiazol-2-ylmethyl)morpholine
N-methyl-2-(methylamino)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-4-carboxamide
N-({8-[(9-ethyl-9H-carbazol-3-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
(2E)-N-({7-[5-(methoxymethyl)furan-2-carbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-phenylprop-2-enamide
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-2-methoxybenzamide
1-(2-cyanobenzoyl)-4-phenoxypiperidine-4-carboxylic acid
methyl (2S,4R)-4-[2-chloro-5-(trifluoromethyl)benzamido]-1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidine-2-carboxylate
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[(3,5-dimethylphenyl)methyl]piperidine-3,5-dicarboxamide
2-(4-chlorophenyl)-4-(3-methoxypyridine-2-carbonyl)morpholine
1-(4-{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
5-(2H-1,3-benzodioxol-5-yl)-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2,4-triazin-3-amine
3-hydroxy-3-({[(2-methylphenyl)methyl]amino}methyl)-1-(3-phenylpropyl)piperidin-2-one
N-(4-fluoro-2-methylphenyl)-4-[(methylsulfanyl)methyl]piperidine-1-carboxamide
4-{2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidine-5-carbonyl}-3-ethylpiperazin-2-one
1-(1-ethylpiperidin-4-yl)-3-(4-phenoxybenzoyl)piperidine
(3aS,6aR)-3-[2-(piperidin-1-yl)ethyl]-5-(9H-purin-6-yl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
6-methoxy-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidin-4-amine
methyl 1-[6-(3-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidine-2-carboxylate
2-(dimethyl-1,3-thiazol-5-yl)-1-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
({4-ethyl-5-[1-(4-methylpiperidine-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-(4-methyl-1H-imidazol-5-yl)-4-(thiophen-2-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-tert-butyl-2-[5-(6-methylpyridin-2-yl)-4-phenyl-1H-imidazol-1-yl]acetamide
1-[4-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
4-acetyl-N-[2-chloro-5-(2-methoxyacetamido)phenyl]piperazine-1-carboxamide
2-[3-(2-fluorophenyl)-1H-pyrazol-1-yl]-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
1-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}-4-(2-phenylethyl)piperazine
2-[(3,4-difluorophenyl)methyl]-8-(1H-imidazol-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
6-methyl-1-{3-oxo-3-[3-(pyridin-2-yl)azetidin-1-yl]propyl}-1,2-dihydropyridin-2-one
methyl 9-[(4-fluorophenyl)methoxy]-7-oxo-3-(2-phenylethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-methyl-2-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]quinoline
3-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-[2-(propan-2-ylsulfanyl)phenyl]urea
3-butyl-1-methyl-4-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]piperazin-2-one
1-(2,3-dihydro-1H-inden-2-yl)-4-{[3-(pyrazin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
N-[(1S,2R)-2-aminocyclobutyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-2-(3-phenylpiperidin-1-yl)pyrimidine
N-(1-propyl-1H-1,2,3-triazol-4-yl)spiro[indene-1,4'-piperidine]-1'-carboxamide
4-[(2-chloro-4-fluorophenyl)methyl]-6-methoxy-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(3-fluorophenyl)methyl]piperazine
N-methyl-2-oxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroquinoline-4-carboxamide
5-butyl-1'-(3-ethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
ethyl 1-[2-(diethylamino)acetyl]-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
4-[3-(2-hydroxyethyl)-4-[(4-methylphenyl)methyl]piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]-6-ethyl-2-methylquinoline
N-(cyclopropylmethyl)-N-propyl-2-(pyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N3-cyclohexyl-N5-[2-(3-fluorophenyl)ethyl]-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[(1-propyl-1H-pyrazol-4-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
1-cyclopentyl-4-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1,4-diazepane
1-(6-ethyl-2-methylpyrimidin-4-yl)-N-[3-(4-methoxyphenyl)propyl]piperidin-4-amine