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N-(2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}phenyl)butanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2-methoxyethyl)-N-methyl-1,3-oxazole-4-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-(1-phenylcyclopropyl)benzamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
1-cyclopentyl-N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-4-[2-(thiophen-3-yl)acetyl]-1,4-diazepan-2-one
1-[(2-fluorophenyl)methyl]-N-{[3-(methylsulfanyl)phenyl]methyl}piperidin-3-amine
1-methanesulfonyl-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,4-diazepane
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
6-methoxy-1-methyl-3-[4-phenyl-1-(1H-1,2,4-triazol-5-ylmethyl)-1H-imidazol-5-yl]-1H-indole
2-(3-chloro-5-methoxybenzoyl)-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)but-3-enamide
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(3-phenylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(oxan-4-yl)piperazin-2-yl}ethan-1-ol
2-{2-[4-(2-methylphenyl)piperazin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
1-(cyclohexylmethyl)-5-[4-(pyridin-3-ylmethyl)piperazine-1-carbonyl]piperidin-2-one
5-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyridine-2,4-diol
1-[6-(2-propyl-1H-imidazol-1-yl)-1,2,3,4-tetrahydroquinolin-1-yl]ethan-1-one
1-(3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)azepane
2-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]pyridin-3-ol
3-(3-methoxypyridin-2-yl)-5-[2-(piperidin-2-yl)ethyl]phenol
4-{1-[2-(dimethylamino)benzoyl]piperidin-3-yl}benzoic acid
2-[({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)amino]-6-methylpyridine-3-carbonitrile
2-(2-methoxyquinoline-4-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(pyrazin-2-yl)ethyl]amino}methyl)piperidin-2-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]benzamide
1-{3-fluoro-8-methylimidazo[1,2-a]pyridine-2-carbonyl}azocane
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-5-methyl-1-[(methylcarbamoyl)methyl]-1H-pyrazole-3-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[2-(diethylamino)ethyl]-N-methylpropanamide
(3R,4R)-1-[(4,5-dimethylfuran-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
methyl 1-[(3S,5S)-1-(furan-3-ylmethyl)-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
6-methyl-N-(pyridin-4-ylmethyl)-2-(pyrrolidin-1-yl)pyrimidin-4-amine
1-cyclohexyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}piperidine-3-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(1R,2R)-N-(furan-2-ylmethyl)-2-phenyl-N-(prop-2-en-1-yl)cyclopropane-1-carboxamide
1-(6-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}pyridazin-3-yl)azepane
1-[3-(azepan-1-yl)propanoyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-(1,4-dioxan-2-ylmethyl)-N,3,6-trimethyl-1-benzofuran-2-carboxamide
1-cyclohexyl-N3-[2-(2-methoxyphenyl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(dimethylamino)ethyl]-5-(3-methyl-1H-pyrazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
5-(phenoxymethyl)-N-(1-propylcyclopropyl)-1H-pyrazole-3-carboxamide
5-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]-2,1,3-benzothiadiazole
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]acetamide
1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-(2-{[5-(methoxymethyl)furan-2-yl]formamido}ethyl)pyridine-3-carboxamide