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2-{1-methyl-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(4-ethylphenyl)-3-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}urea
1-(1H-indole-2-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1-(5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carbonyl)-1,2,3,6-tetrahydropyridine
3-methyl-4-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}-1,2,5-oxadiazole
2-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}benzoic acid
N-tert-butyl-2-[6-(dimethylamino)pyridazin-3-yl]benzene-1-sulfonamide
2-methoxy-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)acetamide
2-methyl-4-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
N-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-(4H-1,2,4-triazol-4-yl)benzamide
6-{1,4-diazabicyclo[3.2.2]nonan-4-yl}-2-(pyrrolidin-1-yl)pyrimidin-4-amine
5-[(4-benzyl-3,5-dimethyl-1H-pyrazol-1-yl)methyl]-3-(cyclopropylmethyl)-1,2,4-oxadiazole
1-[2-(4-fluorophenyl)ethyl]-5-{2-[(2-methoxyethyl)amino]ethyl}pyrrolidin-2-one
methyl 3-[(2,5-dimethylphenyl)methyl]-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-{1-[2-(2-fluorophenyl)ethyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)pyrimidine
1-(cyclohexylmethyl)-5-[(2-methoxyethyl)(methyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]pyrazine-2-carboxamide
N-[(4-chlorophenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-ethyl-1-methyl-N-({3-methyl-7-[2-(thiophen-3-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1H-pyrazole-5-carboxamide
(cyclohex-3-en-1-ylmethyl)(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidine
[(3R,4R)-1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]cyclopropanesulfonamide
methyl 2-[(5-benzenesulfonamido-1-ethyl-2-methyl-1H-1,3-benzodiazol-7-yl)formamido]acetate
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(3-methoxypropyl)-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
1-(furan-2-ylmethyl)-N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}piperidine-4-carboxamide
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-(furan-2-ylmethyl)-1-(1-hydroxybutan-2-yl)urea
5-ethyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-1,2-oxazole-3-carboxamide
methyl 4-{4-[(4aS,8aR)-decahydroisoquinolin-2-ylmethyl]-5-methyl-1,3-oxazol-2-yl}benzoate
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}pyrrolidine-2-carboxamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-ethoxyacetamide
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-{2-oxo-1'-[(2E)-3-phenylprop-2-en-1-yl]-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
(2R,6R)-10-methoxy-4-[(4-methyl-1H-imidazol-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-methyl-5-[4-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
[5-(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]methanol
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(3-methoxyphenyl)methyl]benzamide
6-[(3S,4S)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-[4-(2H-1,3-benzodioxol-5-yl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(1,2-oxazol-3-ylmethyl)acetamide
1-[(2-chlorophenyl)methyl]-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-(4-{[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N-[2-(furan-2-yl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
3-(2-fluorophenyl)-3-{2-[4-(4-hydroxyphenyl)piperazin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)pyrrolidine-2,5-dione
5-(2-fluorophenoxymethyl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-pyrazole-3-carboxamide
6-chloro-N-[(1-methylpyrrolidin-3-yl)methyl]-2-oxo-2H-chromene-3-carboxamide
9-(4-methylpyrimidine-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
ethyl 4-({[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]carbamoyl}amino)piperidine-1-carboxylate
N-[1,3-dihydroxy-2-(hydroxymethyl)propan-2-yl]-3-{[(4-methylphenyl)methyl]amino}benzamide
(4aS,8aR)-1-(3-aminopropyl)-6-[2-(2-oxopyrrolidin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one