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2-[4-(2-methyl-1,3-benzoxazole-6-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-methyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)-N-[2-(piperidin-1-yl)ethyl]propanamide
2-methoxy-5-[(1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octan-6-yl)methyl]phenol
2-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-6-methyl-4H-pyran-4-one
N-[(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]-4-fluorobenzamide
6-methoxy-2-oxo-N-(1,2,3,4-tetrahydroquinolin-1-yl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-methyl-1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-4-(2-methylphenyl)piperazine
1-cycloheptyl-4-{[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]amino}pyrrolidin-2-one
2-(5-acetylthiophen-3-yl)-1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]ethan-1-one
3-(4-methylphenoxymethyl)-1-(5-propyl-1,2-oxazole-4-carbonyl)piperidine
8-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(isoquinolin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[(2-chlorophenyl)methyl]-2-hydroxy-N-(propan-2-yl)pyridine-3-carboxamide
4-(2-ethoxyphenyl)-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{2-chloro-4-[(4-cyclopentyl-3-oxopiperazin-1-yl)methyl]phenoxy}acetamide
2-[2-(6-hydroxy-1,4-oxazepan-4-yl)-4-(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
2-(2,6-difluorophenyl)-N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)acetamide
(2R,3S,6R)-5-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
2-amino-4-(3-hydroxy-4-methoxyphenyl)-5-methyl-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
3-(3-fluoro-4-phenylbenzoyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidine
6-(2-chlorophenyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}imidazo[2,1-b][1,3]thiazole
1-(morpholin-4-yl)-3-[3-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
4-(2H-1,3-benzodioxol-5-ylmethyl)-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
3-propyl-N,N-bis(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
7-(cyclopropylmethyl)-2-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
methyl 3-acetamido-1-ethyl-5-[(thiophen-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{2-[1-(3,4-difluorophenyl)-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
N-{4-[(4-{1-[(2,3-dimethoxyphenyl)methyl]-4-methyl-2,5-dioxoimidazolidin-4-yl}piperidin-1-yl)methyl]phenyl}acetamide
N-[1-({[2-(1H-indol-1-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-{1-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1H-imidazol-2-yl}-2-ethyl-4-methyl-1H-imidazole
N-[(2-fluorophenyl)methyl]-4-(4-{[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)benzamide
2-(azepan-1-yl)-N-({1-[(2E)-2-methylbut-2-en-1-yl]pyrrolidin-3-yl}methyl)-2-oxoacetamide
6-[(3-methoxyphenyl)methoxy]-4-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-1-(2-phenylethyl)-1,4-diazepan-2-one
N4-methyl-N4-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-(propan-2-yl)pyrimidine-2,4-diamine
methyl 3-{[1-(cyclopropylmethyl)-5-(4-fluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]propanamide
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyridazine
1-{5-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-3-yl)propan-1-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(methylsulfanyl)acetamide
3-(4-phenoxybenzoyl)-1-(thiophene-3-carbonyl)piperidine
(2S,4S)-1-cyclopentyl-4-(2,5-dimethylfuran-3-amido)-N,N-diethylpyrrolidine-2-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(2-methyl-1,3-thiazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-[1-(2-fluorophenyl)piperidin-4-yl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
N-[1-(2-chlorophenyl)-5-oxopyrrolidin-3-yl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[(3S,5S)-1-(cyclopropylmethyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-4-methyl-1H-imidazole-2-carboxamide
{4-benzyl-1-[(3-methylphenyl)methyl]piperidin-4-yl}methanol