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1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-methyl-2-(1-methyl-1H-indol-3-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
1-(4-fluorophenyl)-N-[2-(1H-indol-1-yl)ethyl]cyclopropane-1-carboxamide
N-[2-(2-fluorophenyl)-1-[1-(quinoxalin-5-ylmethyl)piperidin-4-yl]ethyl]-N,2-dimethylfuran-3-carboxamide
({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)(methyl)[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]amine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(3-fluorophenyl)piperidine
3-chloro-6-[(3S,4R)-3-acetamido-4-propylpyrrolidin-1-yl]pyridine-2-carboxylic acid
2-(pyridin-4-yl)-5-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]pyrimidin-4-ol
5-[1-(naphthalene-2-carbonyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
5-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
3-{[(furan-3-ylmethyl)(methyl)amino]methyl}-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
3-methoxy-2-(4,5,6,7-tetramethyl-1H-1,3-benzodiazol-2-yl)phenol
4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
2-(2-{[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-(2-fluoro-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)ethan-1-one
(2R)-2-amino-2-phenyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
1-{2-[2-(3,4-dimethoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-ethyl-N-(2-methylprop-2-en-1-yl)piperidine-3-carboxamide
1-[(3-{[2-(3-methoxyphenyl)azetidin-1-yl]methyl}phenyl)methyl]-1H-pyrazole
8-methyl-3-[1-(3-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
6-[(4-benzylpiperidin-1-yl)methyl]-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
1-(3-acetyl-1H-pyrazole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-hydroxy-2-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}quinoline-6-carboxamide
(1R,9aR)-1-{[bis(furan-2-ylmethyl)amino]methyl}-octahydro-1H-quinolizin-1-ol
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3,3-dimethylbutan-1-one
(3aS,6aS)-5-(4-hydroxy-6-oxo-1-phenyl-1,6-dihydropyridazine-3-carbonyl)-N,N-dimethyl-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
5-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
1-(2H-1,3-benzodioxol-5-yl)-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
5-(2-methylpropyl)-3-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2-oxazole
4-[4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-(2-aminoethyl)-N,5,6-trimethyl-N-[2-(pyridin-2-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-1-(2-methoxyethyl)-1-(pyridin-3-ylmethyl)urea
N-ethyl-N-methyl-3-oxo-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecane-9-sulfonamide
2-amino-6-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}pyrimidin-4-ol
N,5-dimethyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-4-carboxamide
2-chloro-5-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)carbamoyl}amino)-N,N-dimethylbenzamide
N-(4-{4-[(dicyclopropylmethyl)amino]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
[(2S)-1-[2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]pyrrolidin-2-yl]methanol
3-[3-(4-aminopiperidin-1-yl)-3-oxopropyl]-3-benzyl-1-methyl-2,3-dihydro-1H-indol-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-benzyl-N,1-dimethyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[(3-chloro-2,6-difluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
methyl({[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}){[3-(trifluoromethyl)phenyl]methyl}amine
[1-(ethylsulfanyl)propan-2-yl]({imidazo[1,2-a]pyridin-2-ylmethyl})amine
1-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]azetidin-3-ol
N-{2-[cyclopentyl(methyl)amino]ethyl}-N,2,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-(3-methylphenoxy)-1-(1H-pyrrole-2-carbonyl)piperidine-4-carboxylic acid
2-methoxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methylquinoline-4-carboxamide
N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
methyl 3-(2,3-dihydro-1,4-benzodioxine-6-sulfonamido)-5-(acetamidomethyl)benzoate
(4aS,7aR)-1-[(3-methoxyphenyl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione