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N-[2-(3,5-dimethylphenoxy)ethyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{2-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[4-(4-{[1-(1,3-thiazol-5-yl)propan-2-yl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
2-{[2-(benzyloxy)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
(3S,4S)-1-[(4-cyanophenyl)methyl]-4-cyclopropylpyrrolidine-3-carboxylic acid
2-[3-(3,4-dimethoxyphenyl)-1H-pyrazol-1-yl]-N-(1-methyl-1H-1,2,3-triazol-4-yl)acetamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]piperidine-3-carboxamide
2-(3-hydroxypropyl)-8-(pyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-{[2-(1H-imidazol-1-yl)ethyl]sulfamoyl}-N-[(3-methyloxetan-3-yl)methyl]benzamide
1-(cyclohex-3-ene-1-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
4-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2-propylpyridine
1-(7-chloro-2-methylquinoline-4-carbonyl)-3-ethylpiperidine-3-carboxylic acid
3-(prop-2-en-1-yl)-1-(thiophen-2-ylmethyl)piperidine-3-carboxylic acid
methyl 2-[4-(2-methoxyethyl)-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetate
(4aR,8aS)-1-[(4-methoxyphenyl)methyl]-6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
3-[(methylsulfanyl)methyl]-5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-1,2,3-thiadiazole-4-carboxamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-methylpiperazine
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
(3R,4R)-3-methyl-1-[2-(methylamino)pyridine-4-carbonyl]-4-(oxan-4-yl)piperidin-4-ol
4-(4-fluoro-2-methylbenzoyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(1R,7S)-3-(3-methylbutyl)-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-cyclopropyl-1H-pyrrole-2-carboxamide
7-(3-chlorophenyl)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4R)-4-benzamido-N,N-diethyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
1-[(2-fluorophenyl)methyl]-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,4-diazepane
ethyl 1-[6-(4-methylthiophen-2-yl)-3-[(1,2-oxazol-3-ylmethyl)carbamoyl]pyridin-2-yl]piperidine-4-carboxylate
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)cyclopropanesulfonamide
{3-[5-(1-methyl-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]phenyl}methanol
ethyl({[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})(pyridin-4-ylmethyl)amine
ethyl 1-(dimethyl-1,3-thiazole-5-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-[4-(3-methoxypyrazin-2-yl)-1H-pyrazol-1-yl]-N-(2-propyl-2H-1,2,3-triazol-4-yl)acetamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](ethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-amino-3-ethyl-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[(3-methoxyphenyl)amino]-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)butanamide
1-(2-methylphenyl)-4-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1,4-diazepane
methyl({[5-(oxan-2-yl)thiophen-2-yl]methyl})[2-(pyridin-2-yl)ethyl]amine
3-benzoyl-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidine
3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]urea
4-(5-chloro-2-hydroxybenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1,3-oxazole-4-carboxamide
(2E)-3-(3-fluorophenyl)-N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)prop-2-enamide
4-[(diethylamino)methyl]-5-ethyl-N-[2-(3-hydroxypiperidin-1-yl)ethyl]furan-2-carboxamide
N-({7-[(2,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
2-(2-{[1-(pyrazin-2-yl)piperidin-4-yl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
5-(benzyloxy)-2-({1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}methyl)phenol
6-methyl-2-{[2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]amino}-3,4-dihydropyrimidin-4-one
2-amino-6-cyclopropyl-4-[5-(oxolan-2-yl)thiophen-2-yl]pyridine-3-carbonitrile
(3S,4S)-1-cyclopropanecarbonyl-4-(naphthalen-2-yl)piperidin-3-ol
2-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one