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4-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-2-(6-methoxynaphthalen-2-yl)morpholine
(2S)-2-amino-1-{4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}propan-1-one
methyl (1S,3S,3aR,6aS)-3-(3-cyanophenyl)-5-methyl-4,6-dioxo-1-phenyl-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
4-{2-[(1-acetylpiperidin-4-yl)oxy]-5-chlorobenzoyl}-3,3-dimethylpiperazin-2-one
N,5,6-trimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
N3-[(1-hydroxycyclohexyl)methyl]-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-N-({8-[(6-methylpyridin-2-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-thiazole-4-carboxamide
N-(1-{1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1-dimethyl-1H-pyrazole-3-carboxamide
3-(3,4-dimethoxyphenyl)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-methoxy-5-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenol
2-[4-(propan-2-yloxy)phenyl]-2-(4-propyl-1,4-diazepan-1-yl)acetic acid
(3S,4R)-1-(2-aminopyridine-4-carbonyl)-3-benzyl-4-methylpiperidin-4-ol
5,6-dimethyl-3-(2,2,6,6-tetramethylpiperidin-4-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-ethoxy-4-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}phenol
2-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-2,3-dihydro-1H-isoindole
N-cyclopropyl-2-(dimethylamino)-2-(4-methylphenyl)-N-(pyridin-4-ylmethyl)acetamide
{3-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl}methanamine
2,4-dimethyl-N-{4-[4-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)piperidin-1-yl]phenyl}benzamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(2-oxoazepan-1-yl)propanamide
4-{[2-(hydroxymethyl)phenyl]methyl}-N-[3-(methylcarbamoyl)phenyl]piperazine-1-carboxamide
N-{[4-(2-methylpropoxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)benzamide
1-[2-(dimethylamino)ethyl]-4-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]pyrrolidin-2-one
6-[(4-fluorophenyl)methoxy]-4-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1-(propan-2-yl)-1,4-diazepan-2-one
6-(piperidin-1-yl)-N-[2-(pyridin-3-yloxy)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
3-[2-(2,4-difluorophenyl)ethyl]-1-(4-methyl-1,3-thiazole-5-carbonyl)piperidine
5-(2-chloro-5-methylphenyl)-3-(propan-2-yl)-1,2,4-oxadiazole
3-[1-(5-hydroxypentyl)-4-phenyl-1H-imidazol-5-yl]phenol
N-[(3R,4S)-4-(4-methoxyphenyl)-1-[2-oxo-2-(piperidin-1-yl)ethyl]pyrrolidin-3-yl]acetamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-ethyl-1H-pyrazole-4-carboxamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine-4-carboxylate
6-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}pyrazolo[1,5-a]pyrimidine-3-carboxylic acid
4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{[1-(3-hydroxypyridine-2-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
N-ethyl-2-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}acetamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-(3-chlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-benzoyl-N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]piperidin-4-amine
3-(3-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-1H-indol-1-yl)propanamide
3-{benzyl[(5-ethylpyridin-2-yl)methyl]amino}-2-methylpropan-1-ol
2-[N-(3-fluorophenyl)methanesulfonamido]-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]-N'-(4-methylphenyl)propanediamide
1-[(3-methoxyphenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-1-(propan-2-yl)-1H-1,3-benzodiazole
N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methoxyacetamide
(2S,4R)-4-amino-N,N-diethyl-1-(2-fluoro-4-methylbenzenesulfonyl)pyrrolidine-2-carboxamide
4-methyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1,3-thiazole-5-carboxamide
1-(diethylamino)-3-[2-methoxy-4-({[3-(2-methyl-1H-imidazol-1-yl)propyl]amino}methyl)phenoxy]propan-2-ol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)but-3-enamide
5-[2-(benzenesulfonyl)ethyl]-2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine