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N-{1-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}propanamide
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-cyclopentylpiperazin-2-yl]ethan-1-ol
N-[2-(4-methylmorpholin-2-yl)ethyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-{1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}piperidin-3-ol
methyl 5-[(4-hydroxy-4-methylpentan-2-yl)amino]-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
(8R,9aS)-8-hydroxy-2-[2-(1H-indol-3-yl)ethyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
4-(cyclopropylmethyl)-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
(3S,9aR)-3-[(1R)-1-hydroxyethyl]-8-[(5-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
methyl 3-{[1-(cyclopropylmethyl)-5-(2-methoxybenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
7-(cyclopropylmethyl)-2-(2-methyl-1-benzofuran-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(3-fluorophenyl)methyl]-4-[3-(methylsulfanyl)butyl]piperazine
2,2-dimethyl-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}propanamide
1-[4-(hydroxymethyl)-4-(2-phenylethyl)piperidin-1-yl]-2-(pyridin-4-ylsulfanyl)ethan-1-one
1-{[5-(1-cyclopentanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}azepane
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(1,2-oxazol-5-ylmethyl)acetamide
5-acetyl-N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}thiophene-3-carboxamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-1-(2-phenylethyl)piperidine
1-(2-{4-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-1H-1,2,3-triazol-1-yl}ethyl)piperazine
N-(1-methylpiperidin-4-yl)-5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[2-(3-methoxyphenyl)ethyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-(1-phenylcyclopropyl)acetamide
{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
N3-[2-(2-fluorophenyl)ethyl]-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(cyclopropylmethyl)-9-[3-(4-hydroxyphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(2-methoxyacetamido)-1-(2-phenylethyl)-N-[(1S)-1-phenylethyl]-1H-1,3-benzodiazole-7-carboxamide
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-2-(2-methoxyethyl)pyrimidine
(2S,4S,5R)-2-ethyl-4-[(3-hydroxypropyl)(methyl)carbamoyl]-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
4-hydroxy-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(phenoxymethyl)pyrimidine-5-carboxamide
1-(oxan-4-yl)-4-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperazine
2-{4-[2-(2-phenylethyl)pyrrolidine-1-carbonyl]phenoxy}acetamide
5-(3-methyl-1,2,4-oxadiazol-5-yl)-2-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}pyridine
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-(4-methylphenoxy)piperidine-4-carboxylic acid
N-(4-{1-[(2S)-1-hydroxy-4-methylpentan-2-yl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
(3R,4R)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-(2,4-dichlorophenoxy)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}acetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
3-(2-ethyl-1H-imidazol-1-yl)-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)propan-1-one
3-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-[3-(1,3-thiazol-4-yl)phenyl]urea
3-[2-({1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}amino)propyl]-3,4-dihydroquinazolin-4-one
(1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(pyridin-3-yl)methanol
1-(2-methanesulfonylethyl)-4-(3-methoxy-5-methylthiophene-2-carbonyl)piperazine
1-[(2-chlorophenyl)methyl]-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1H-1,2,3-triazole-4-carboxamide
5-{1-[2-(3,4-dimethoxyphenyl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
1-[4-(3-methylpiperidine-1-carbonyl)phenyl]-3-[(5-methylpyrazin-2-yl)methyl]urea
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)thieno[2,3-d]pyrimidin-4-amine
4-(2,4-dioxoimidazolidin-1-yl)-N-[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]benzamide